Compile Data Set for Download or QSAR
maximum 50k data
Found 209 with Last Name = 'höglund' and Initial = 'i'
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196109((2,3-dimethylquinolin-4-yl)-[4-(octahydro-2H-pyrid...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM508526(N-((S)-1-(3-(3-chloro-4-cyano-2-methylphenyl)-1H-p...)
Affinity DataKi:  3nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309987(N-((S)-1-(3-(3-chloro-4-cyano-2-methylphenyl)-1H-p...)
Affinity DataKi:  3nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196123(CHEMBL218675 | {2-methyl-4-[4-(3,3,4-trimethylpipe...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196117(1-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]-2...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196142(CHEMBL218457 | [4-(3,4-dimethylpiperazin-1-yl)phen...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196132(CHEMBL217203 | [4-(3,4-dimethylpiperazin-1-yl)phen...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196139((3-methylquinolin-4-yl)-[4-(3,3,4-trimethylpiperaz...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196107(CHEMBL216464 | {7-chloro-4-[4-(3,3,4-trimethylpipe...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309973((S)-N-(1-(3-(4-cyano-3-methylphenyl)-1H-pyrazol-1-...)
Affinity DataKi:  6nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309973((S)-N-(1-(3-(4-cyano-3-methylphenyl)-1H-pyrazol-1-...)
Affinity DataKi:  6nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196118(CHEMBL268217 | {4-[4-(3,3,4-trimethylpiperazin-1-y...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196146(CHEMBL217177 | [4-(3,4-dimethylpiperazin-1-yl)phen...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196129(CHEMBL214996 | {4-[4-(3,4-dimethylpiperazin-1-yl)p...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196145((R)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7,...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309982((S)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  8nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309982((S)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  8nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50418050(CHEMBL1689423)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196125((R)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7-...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196131(CHEMBL217202 | [4-(3,4-dimethylpiperazin-1-yl)phen...)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196147((3-ethyl-2,8-dimethylquinolin-4-yl)-[4-(4-methyl-[...)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196126((R)-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196116((R)-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM508530((R)-N-(2-(3-(4-cyano-3,5-difluorophenyl)-1H-pyrazo...)
Affinity DataKi:  12nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309988((S)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  12nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309990((R)-N-(2-(3-(4-cyano-3,5-difluorophenyl)-1H-pyrazo...)
Affinity DataKi:  12nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309988((S)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  12nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309981((S)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  13nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM508521((S)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  13nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM508519(N-((S)-1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  14nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309979(N-((S)-1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  14nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM508534((S)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  14nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309995((S)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  14nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196113(CHEMBL262901 | [4-(3,4-dimethylpiperazin-1-yl)phen...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309976((S)-3-acetyl-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-p...)
Affinity DataKi:  16nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196120(CHEMBL216727 | [4-(3,4-dimethylpiperazin-1-yl)phen...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309992((S)-N-{1-[3-(3-Chloro-4-cyano-5-fluorophenyl)-1H-p...)
Affinity DataKi:  16nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309992((S)-N-{1-[3-(3-Chloro-4-cyano-5-fluorophenyl)-1H-p...)
Affinity DataKi:  16nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309976((S)-3-acetyl-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-p...)
Affinity DataKi:  16nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309983(N-((R)-1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  17nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM508523((S)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  17nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309980(N-(2-(3-(4-cyano-3-methylphenyl)-1H-pyrazol-1-yl)e...)
Affinity DataKi:  18nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309980(N-(2-(3-(4-cyano-3-methylphenyl)-1H-pyrazol-1-yl)e...)
Affinity DataKi:  18nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309993((S)-N-(1-(3-(3-chloro-4-cyano-5-fluorophenyl)-1H-p...)
Affinity DataKi:  25nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196136((3-ethyl-2-methylquinolin-4-yl)-[4-(4-methylpipera...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309993((S)-N-(1-(3-(3-chloro-4-cyano-5-fluorophenyl)-1H-p...)
Affinity DataKi:  25nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309978(N-(2-(3-(3,4-dicyanophenyl)-1H-pyrazol-1-yl)ethyl)...)
Affinity DataKi:  27nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309978(N-(2-(3-(3,4-dicyanophenyl)-1H-pyrazol-1-yl)ethyl)...)
Affinity DataKi:  27nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196135(Acridin-9-yl-[4-(4-methyl-piperazin-1-yl)-phenyl]-...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Orion

US Patent
LigandPNGBDBM309986((R)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-...)
Affinity DataKi:  29nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 209 total ) | Next | Last >>
Jump to: