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Found 35 with Last Name = 'hacker' and Initial = 'm'
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50495103(CHEMBL3105243)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]WIN35428 from human DAT after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50495101(CHEMBL1945251)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]Nisoxetine from human SERT after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50495101(CHEMBL1945251)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]WIN35428 from human DAT after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50495103(CHEMBL3105243)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]Nisoxetine from human SERT after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM22166(3-(4-iodophenyl)tropane-2-carboxylic acid methyl e...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity to DAT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50296782((1R,2S,3S,5S)-methyl 8-((E)-3-iodoallyl)-3-p-tolyl...)
Affinity DataKi:  17nMAssay Description:Binding affinity to DAT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50495101(CHEMBL1945251)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]Imipramin from human NET after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM22166(3-(4-iodophenyl)tropane-2-carboxylic acid methyl e...)
Affinity DataKi:  29nMAssay Description:Binding affinity to SERT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM22166(3-(4-iodophenyl)tropane-2-carboxylic acid methyl e...)
Affinity DataKi:  33nMAssay Description:Binding affinity to NET (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50495102(CHEMBL3105242)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]WIN35428 from human DAT after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50495102(CHEMBL3105242)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]Nisoxetine from human SERT after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50495103(CHEMBL3105243)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]Imipramin from human NET after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50296782((1R,2S,3S,5S)-methyl 8-((E)-3-iodoallyl)-3-p-tolyl...)
Affinity DataKi:  500nMAssay Description:Binding affinity to SERT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50495102(CHEMBL3105242)
Affinity DataKi:  785nMAssay Description:Displacement of [3H]Imipramin from human NET after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50296782((1R,2S,3S,5S)-methyl 8-((E)-3-iodoallyl)-3-p-tolyl...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to NET (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65554(Synthesized Sulfanylacrylonitril Derivatives 5)
Affinity DataIC50:  120nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65548(Synthesized Sulfanylacrylonitril Derivatives 2)
Affinity DataIC50:  260nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65563(Synthesized Sulfanylacrylonitril Derivatives 10)
Affinity DataIC50:  470nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65571(Synthesized Sulfanylacrylonitril Derivatives 18)
Affinity DataIC50:  570nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65565(Synthesized Sulfanylacrylonitril Derivatives 12)
Affinity DataIC50:  800nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65564(Synthesized Sulfanylacrylonitril Derivatives 11)
Affinity DataIC50:  940nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65572(Synthesized Sulfanylacrylonitril Derivatives 19)
Affinity DataIC50:  960nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65568(Synthesized Sulfanylacrylonitril Derivatives 15)
Affinity DataIC50:  1.30E+3nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65573(Synthesized Sulfanylacrylonitril Derivatives 20)
Affinity DataIC50:  1.77E+3nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65562(Synthesized Sulfanylacrylonitril Derivatives 9)
Affinity DataIC50:  1.82E+3nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65569(Synthesized Sulfanylacrylonitril Derivatives 16)
Affinity DataIC50:  2.51E+3nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65567(Synthesized Sulfanylacrylonitril Derivatives 14)
Affinity DataIC50:  4.62E+3nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65577(Synthesized Sulfanylacrylonitril Derivatives 21)
Affinity DataIC50:  1.13E+4nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65558(Synthesized Sulfanylacrylonitril Derivatives 7)
Affinity DataIC50:  1.63E+4nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65570(Synthesized Sulfanylacrylonitril Derivatives 17)
Affinity DataIC50:  2.18E+4nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65551(Synthesized Sulfanylacrylonitril Derivatives 3)
Affinity DataIC50: >3.00E+4nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65552(Synthesized Sulfanylacrylonitril Derivatives 4)
Affinity DataIC50: >1.00E+5nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65556(Synthesized Sulfanylacrylonitril Derivatives 6)
Affinity DataIC50: >1.00E+5nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65578(Synthesized Sulfanylacrylonitril Derivatives 22)
Affinity DataIC50: >1.00E+5nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4-A phosphorylase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Konstanz

LigandPNGBDBM65560(Synthesized Sulfanylacrylonitril Derivatives 8)
Affinity DataIC50: >1.00E+5nMpH: 8.0Assay Description:Dose response curves against Rv2613c with 1 as the substrate for derivatives 5 and 18. 8 nM of Rv2613c were preincubated in buffer (20 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed