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Found 21 with Last Name = 'hadac' and Initial = 'em'
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  0.800nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50072425(2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-...)
Affinity DataIC50:  50nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50181434((S)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-p...)
Affinity DataIC50:  61nMAssay Description:Displacement of [125I-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat CCK receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50072421(2-{3-[3-(3-Benzoyl-phenyl)-ureido]-2,4-dioxo-5-phe...)
Affinity DataIC50:  80nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50072422(2-{3-[3-(3-Benzoyl-phenyl)-ureido]-2,4-dioxo-5-phe...)
Affinity DataIC50:  160nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50072427(1-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl)-2,4-d...)
Affinity DataIC50:  250nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50072420(2-{3-[3-(3-Benzoyl-phenyl)-ureido]-2,4-dioxo-5-phe...)
Affinity DataIC50:  290nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50072424(2-(2,4-Dioxo-5-phenyl-3-{3-[3-(3-trifluoromethyl-3...)
Affinity DataIC50:  310nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50072428(2-{3-[3-(3-Benzoyl-phenyl)-ureido]-2,4-dioxo-5-phe...)
Affinity DataIC50:  350nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50072419(2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-...)
Affinity DataIC50:  390nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50072429(2-(2,4-Dioxo-5-phenyl-3-{3-[3-(3-trifluoromethyl-3...)
Affinity DataIC50:  410nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50072423(2-(2,4-Dioxo-5-phenyl-3-{3-[3-(3-trifluoromethyl-3...)
Affinity DataIC50:  440nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50181435((R)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-p...)
Affinity DataIC50:  470nMAssay Description:Displacement of [125I-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat CCK receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50181433((S)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-p...)
Affinity DataIC50:  490nMAssay Description:Displacement of [125I-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat CCK receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50181436((R)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-p...)
Affinity DataIC50:  710nMAssay Description:Displacement of [125I-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat CCK receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50072426(2-(2,4-Dioxo-5-phenyl-3-{3-[3-(3-trifluoromethyl-3...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of 125I]-D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat cell membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataEC50:  0.00900nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50472278(CHEMBL410965)
Affinity DataEC50:  150nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50472277(CHEMBL438912)
Affinity DataEC50:  280nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50472279(CHEMBL405243)
Affinity DataEC50:  28nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50181434((S)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-p...)
Affinity DataEC50:  150nMAssay Description:Intrinsic agonistic activity at CCK receptor in SD rat at 1uM expressed in pancreatic acinar cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed