Affinity DataKi: 4.30E+3nM ΔG°: -31.9kJ/mole IC50: 1.02E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 3(Bos taurus)
Pohang University Of Science & Technology
Curated by ChEMBL
Pohang University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Binding affinity towards Inositol 1,4,5-trisphosphate receptor was evaluated by the standard competitive binding assay using 1.25 nM [3H]-D-I(1,4,5)P...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 348nMAssay Description:Inhibition of HSP90 using VER-00045864 probe by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of estrogen sulfotransferase (EST) in TLC radiolabel transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 560nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
TargetInositol 1,4,5-trisphosphate receptor type 3(Bos taurus)
Pohang University Of Science & Technology
Curated by ChEMBL
Pohang University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 598nMAssay Description:Binding affinity towards Inositol 1,4,5-trisphosphate receptor was evaluated by the standard competitive binding assay using 1.25 nM [3H]-D-I(1,4,5)P...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 790nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair