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Found 4711 with Last Name = 'haque' and Initial = 'ts'
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076285(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  1.30nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076294(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  1.90nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076291(1-Methyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  2nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076292(1-Methyl-piperidine-4-carboxylic acid {(2S,3S)-3-[...)
Affinity DataKi:  2nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076285(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  3nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119489(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi:  4nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076294(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  4nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119488(CHEMBL143628 | X1-(4-Chloro-phenyl)-1H-pyrazole-3,...)
Affinity DataKi:  4nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076287(1-Methyl-piperidine-4-carboxylic acid [(2S,3S)-3-(...)
Affinity DataKi:  4.10nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076293(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  4.30nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM8019(2-(3-chlorophenoxy)-N-[(2S,3S)-3-hydroxy-4-{N-[2-(...)
Affinity DataKi:  4.30nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076293(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  4.80nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076291(1-Methyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  5.80nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119481(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi:  6nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119483(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi:  8nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076288(CHEMBL284955 | Piperidine-4-carboxylic acid [(2S,3...)
Affinity DataKi:  9nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076292(1-Methyl-piperidine-4-carboxylic acid {(2S,3S)-3-[...)
Affinity DataKi:  9.80nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119485(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  12nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076286(CHEMBL34051 | N-(2-Benzo[1,3]dioxol-5-yl-ethyl)-N-...)
Affinity DataKi:  15nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119490(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  26nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119492(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi:  32nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076287(1-Methyl-piperidine-4-carboxylic acid [(2S,3S)-3-(...)
Affinity DataKi:  58nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM8019(2-(3-chlorophenoxy)-N-[(2S,3S)-3-hydroxy-4-{N-[2-(...)
Affinity DataKi:  63nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076288(CHEMBL284955 | Piperidine-4-carboxylic acid [(2S,3...)
Affinity DataKi:  71nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119487(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi:  91nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076289(CHEMBL32997 | N-((1S,2S)-3-{(2-Benzo[1,3]dioxol-5-...)
Affinity DataKi:  100nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119491(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  138nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076286(CHEMBL34051 | N-(2-Benzo[1,3]dioxol-5-yl-ethyl)-N-...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076290(CHEMBL284151 | N-(2-Benzo[1,3]dioxol-5-yl-ethyl)-N...)
Affinity DataKi:  300nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119484(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  331nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119482(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119486(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119485(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119484(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119486(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119491(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119487(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119490(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119489(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119488(CHEMBL143628 | X1-(4-Chloro-phenyl)-1H-pyrazole-3,...)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119483(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119492(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119481(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119482(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM568223(US11420973, Example 101)
Affinity DataIC50:  0.340nMAssay Description:HEK-Blue™-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducibl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetToll-like receptor 7(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM566998(US11420958, Ex. No. 367)
Affinity DataIC50:  0.370nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetToll-like receptor 7(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM443999(US10660877, Example 588)
Affinity DataIC50:  0.5nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetToll-like receptor 8(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM566897(US11420958, Ex. No. 266)
Affinity DataIC50:  0.5nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetToll-like receptor 8(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM566956(US11420958, Ex. No. 325)
Affinity DataIC50:  0.5nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetToll-like receptor 8(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM566939(US11420958, Ex. No. 308)
Affinity DataIC50:  0.5nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 4711 total ) | Next | Last >>
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