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Found 80 with Last Name = 'harakawa' and Initial = 'h'
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040108(11-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)-ethylsulfa...)
Affinity DataKi:  6.90nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002084(11-(2-Dimethylamino-ethylsulfanyl)-6,11-dihydro-di...)
Affinity DataKi:  9nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040114(CHEMBL336198 | {11-[2-(4-Benzyl-piperidin-1-yl)-et...)
Affinity DataKi:  10nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002088(CHEMBL302005 | [11-(2-Dimethylamino-ethylidene)-6,...)
Affinity DataKi:  11nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040109(3-{11-[2-(4-Benzyl-piperidin-1-yl)-ethylsulfanyl]-...)
Affinity DataKi:  12nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040112(11-[2-(4-Benzyl-piperazin-1-yl)-ethylsulfanyl]-6,1...)
Affinity DataKi:  14nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50175516(CHEMBL372588 | {11-[2-(4-Benzyl-piperidin-1-yl)-et...)
Affinity DataKi:  15nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040110(2-{11-[2-(4-Benzyl-piperidin-1-yl)-ethylsulfanyl]-...)
Affinity DataKi:  17nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040121(11-[2-(4-Phenyl-piperidin-1-yl)-ethylsulfanyl]-6,1...)
Affinity DataKi:  20nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040111(CHEMBL133080 | {11-[2-(4-Benzyl-piperidin-1-yl)-et...)
Affinity DataKi:  20nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040113(11-{2-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-ethylsu...)
Affinity DataKi:  41nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040116(11-(2-Morpholin-4-yl-ethylsulfanyl)-6,11-dihydro-d...)
Affinity DataKi:  42nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040119(11-[2-(4-Phenyl-piperazin-1-yl)-ethylsulfanyl]-6,1...)
Affinity DataKi:  47nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040117(11-{2-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-pi...)
Affinity DataKi:  500nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040115(CHEMBL133778 | Sodium; 11-[2-(4-benzyl-piperidin-1...)
Affinity DataKi:  740nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50227346(CHEMBL319928)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity was measured for Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50227346(CHEMBL319928)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity was measured for Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50227346(CHEMBL319928)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity was measured for Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040815(2-Methylsulfanyl-6,11-dihydro-dibenzo[b,e]oxepine-...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284967(1-[1-(2,6-Dichloro-phenyl)-1H-benzoimidazol-2-yl]-...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284976(1-[1-(2-Chloro-phenyl)-1H-benzoimidazol-2-yl]-3-(2...)
Affinity DataIC50:  18nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284971(1-(2,6-Diisopropyl-phenyl)-3-(1-o-tolyl-1H-benzoim...)
Affinity DataIC50:  19nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284972(1-(2,6-Diisopropyl-phenyl)-3-[1-(2-methoxy-phenyl)...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284979(1-[1-(3-Chloro-phenyl)-1H-benzoimidazol-2-yl]-3-(2...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284973(1-[1-(2-Bromo-phenyl)-1H-benzoimidazol-2-yl]-3-(2,...)
Affinity DataIC50:  22nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040830(2-Bromo-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  23nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040849(5H-Dibenzo[a,d]cycloheptene-5-carboxylic acid (2,6...)
Affinity DataIC50:  25nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040854(11-(2,6-Diisopropyl-phenylcarbamoyl)-2-methyl-6,11...)
Affinity DataIC50:  27nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284965(1-[3-(2-Chloro-phenyl)-3H-imidazo[4,5-b]pyridin-2-...)
Affinity DataIC50:  33nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040828(2-Iodo-6,11-dihydro-dibenzo[b,e]oxepine-11-carboxy...)
Affinity DataIC50:  35nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040831(3-Bromo-10,11-dihydro-5H-dibenzo[a,d]cycloheptene-...)
Affinity DataIC50:  39nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040826(10,11-Dihydro-5H-dibenzo[a,d]cycloheptene-5-carbox...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284978(1-(2,6-Diisopropyl-phenyl)-3-[1-(2-dimethylamino-p...)
Affinity DataIC50:  41nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040855(2-Methyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040851(3-Methyl-10,11-dihydro-5H-dibenzo[a,d]cycloheptene...)
Affinity DataIC50:  55nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040841(2,9-Dibromo-6,11-dihydro-dibenzo[b,e]oxepine-11-ca...)
Affinity DataIC50:  58nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040848(2,3-Dimethyl-6,11-dihydro-dibenzo[b,e]oxepine-11-c...)
Affinity DataIC50:  64nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284970(1-(2,6-Diisopropyl-phenyl)-3-(1-phenyl-1H-benzoimi...)
Affinity DataIC50:  66nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284974(1-(2,6-Diisopropyl-phenyl)-3-[1-(2-trifluoromethyl...)
Affinity DataIC50:  72nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040843(2-Bromo-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  74nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040840(7-Bromo-5,11-dihydro-10-oxa-1-aza-dibenzo[a,d]cycl...)
Affinity DataIC50:  78nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040824(6,11-Dihydro-dibenzo[b,e]oxepine-11-carboxylic aci...)
Affinity DataIC50:  94nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284969(1-(2,6-Diisopropyl-phenyl)-3-[1-(2-methyl-pyridin-...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50284975(1-[1-(3-Chloro-pyridin-2-yl)-1H-benzoimidazol-2-yl...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibitory activity towards acyl CoA cholesterol acyltransferase (ACAT) of cholesterol-fed rabbits by the displacement of [14C]-oleolyl-CoAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040822(4-Bromo-2-methyl-6,11-dihydro-dibenzo[b,e]oxepine-...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040829(2-Methyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  110nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040817(9-Bromo-2-methyl-6,11-dihydro-dibenzo[b,e]oxepine-...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040814(2-Ethyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040837(2-Methoxy-6,11-dihydro-dibenzo[b,e]oxepine-11-carb...)
Affinity DataIC50:  140nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040818(2-Chloro-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  150nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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