Affinity DataIC50: 2.53nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.62nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
Affinity DataIC50: 3.16nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 4.45nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
Affinity DataIC50: 14.8nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
Affinity DataIC50: 16.9nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 17.7nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 20.3nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 23.8nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
Affinity DataIC50: 25.9nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
Affinity DataIC50: 28.5nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
Affinity DataIC50: 32.6nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 32.7nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
Affinity DataIC50: 65.5nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
Affinity DataIC50: 87.1nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
Affinity DataIC50: 106nMAssay Description:Inhibition of recombinant EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Mus musculus)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant mouse ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
Affinity DataIC50: 190nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of ACSL1 (unknown origin) assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by ...More data for this Ligand-Target Pair
TargetLong-chain-fatty-acid--CoA ligase 1(Homo sapiens)
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Shionogi Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant human ACSL1 assessed as reduction in acetyl-coA prodution incubated for 90 mins in presence of Coenzyme A, ATP and MgCl2 by...More data for this Ligand-Target Pair
Affinity DataIC50: 270nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase (b-TNAP, c-IAP purchased from Calzyme Laboratories, Inc. USA) inhibition assay of different cyclic sulfonamides was performed us...More data for this Ligand-Target Pair