Affinity DataKi: 0.690nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.730nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.770nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.940nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the presence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 1.46nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 2.13nMAssay Description:Binding affinity at human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Competitive inhibition of human NPP1 using p-Nph-5'-TMP as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of human NPP1 using p-Nph-5'-TMP as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the presence of GTPMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Competitive inhibition of human NPP1 using p-Nph-5'-TMP as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of human NPP1 using p-Nph-5'-TMP as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of human NPP1 using p-Nph-5'-TMP as substrateMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Competitive inhibition of human NPP1 using p-Nph-5'-TMP as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Competitive inhibition of human NPP1 using p-Nph-5'-TMP as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Inhibition of human NPP1 using p-Nph-5'-TMP as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the presence of GTPMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Competitive inhibition of human NPP1 using p-Nph-5'-TMP as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Inhibition of human NPP1 using p-Nph-5'-TMP as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the presence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the presence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Non-competitive inhibition of human NPP1 expressed in African green monkey COS7 cells using p-Nph-5'-TMP as substrate after 60 mins by Dixon plot ana...More data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the presence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 102nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
Affinity DataKi: 112nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 114nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the presence of GTPMore data for this Ligand-Target Pair