Affinity DataIC50: 14nMAssay Description:Inhibition of [125I]endothelin-1 [ET-1] binding to endothelin A receptor (ETA) of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Displacement of [125I]-ET-1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Displacement of [125I]-ET-1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of [125I]-endothelin-3 [ET-3] binding to endothelin B receptor (ETB) of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of [125I]endothelin-1 [ET-1] binding to endothelin A receptor (ETA) of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]-ET-1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of [125I]-endothelin-3 [ET-3] binding to endothelin B receptor (ETB) of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Binding affinity against endothelin receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 930nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of [125I]endothelin-1 [ET-1] binding to endothelin A receptor (ETA) of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of [125I]-endothelin-3 [ET-3] binding to endothelin B receptor (ETB) of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of [125I]endothelin-1 [ET-1] binding to endothelin A receptor (ETA) of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of [125I]-endothelin-3 [ET-3] binding to endothelin B receptor (ETB) of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of [125I]-endothelin-3 [ET-3] binding to endothelin B receptor (ETB) of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of [125I]-endothelin-3 [ET-3] binding to endothelin B receptor (ETB) of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of [125I]endothelin-1 [ET-1] binding to endothelin A receptor (ETA) of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of [125I]-endothelin-3 [ET-3] binding to endothelin B receptor (ETB) of rat cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 9.10E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair