TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.331nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q/T423H mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.427nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M2 receptor expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.437nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 W422A mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.724nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M5 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M5 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M2 receptor expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q/T423H mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M2 receptor expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M2 receptor expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q/T423H mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 W422A mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M2 receptor expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M5 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 W422A mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q/T423H mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q/T423H mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q/T423H mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranes preincubated for 30 mins followed by [3...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M2 receptor expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 5.20nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M2 receptor expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q/T423H mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M5 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M2 receptor expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 W422A mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 6.90nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 W422A mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q/T423H mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M2 receptor expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 8.5nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 8.90nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Inhibition of human CYP2D6 by Lineweaver-Burk plotMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y104A mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of recombinant human FKBP12 expressed in Escherichia coli using succinyl-Ala-Phe-Pro-Phe-4-nitroanilide as substrateMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y104A mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 W422A mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
University Of W£Rzburg
Curated by ChEMBL
University Of W£Rzburg
Curated by ChEMBL