TargetBone morphogenetic protein 1(Homo sapiens (Human))
Glaxosmithkline Pharmaceuticals
Curated by ChEMBL
Glaxosmithkline Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 0.00680nMAssay Description:Binding affinity to BMP1 (unknown origin) using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5,6 TAMRA)-CONH2 as substrate preincubated for 3 hrs followed by subs...More data for this Ligand-Target Pair
Affinity DataKi: 0.0310nMAssay Description:Binding affinity to TLL1 (unknown origin) using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5,6 TAMRA)-CONH2 as substrate incubated for 3.5 hrs followed by subst...More data for this Ligand-Target Pair
Affinity DataKi: 0.0390nMAssay Description:Binding affinity to TLL2 (unknown origin) using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5,6 TAMRA)-CONH2 as substrate incubated for 3.5 hrs followed by subst...More data for this Ligand-Target Pair
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Glaxosmithkline Pharmaceuticals
Curated by ChEMBL
Glaxosmithkline Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:Binding affinity to BMP1 (unknown origin) using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5,6 TAMRA)-CONH2 as substrate preincubated for 3 hrs followed by subs...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.229nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Binding affinity to TLL1 (unknown origin) using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5,6 TAMRA)-CONH2 as substrate incubated for 3.5 hrs followed by subst...More data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity to TLL2 (unknown origin) using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5,6 TAMRA)-CONH2 as substrate incubated for 3.5 hrs followed by subst...More data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Binding affinity was determined for the alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Binding affinity against human Alpha-1D adrenergic receptor (h alpha-1d)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.347nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Binding affinity against human Alpha-1a adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity against human Alpha-2b adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.525nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Binding affinity against human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Binding affinity was determined for the alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.580nMAssay Description:Binding affinity against human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.580nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.840nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity against human Alpha-1a adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity against human Alpha-1a adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.87nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Binding affinity against human Alpha-1a adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
Synaptic Pharmaceutical
Curated by ChEMBL
Synaptic Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity against rat L-type calcium channelMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.19nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.42nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.57nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.88nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity against human Alpha-1a adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Binding affinity against human Alpha-1a adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Binding affinity against human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.58nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.66nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.72nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Binding affinity against human Alpha-1a adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Binding affinity against human Alpha-1a adrenergic receptorMore data for this Ligand-Target Pair