TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 8.80nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 103nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 131nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 165nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 169nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 191nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 198nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 201nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 205nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 224nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 232nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 243nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 387nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 574nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 580nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 655nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 992nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 1.11E+3nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 1.11E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 1.42E+3nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 1.45E+3nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 1.47E+3nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 1.57E+3nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 1.63E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 1.73E+3nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 1.77E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 1.89E+3nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Tennessee
Curated by ChEMBL
University Of Tennessee
Curated by ChEMBL
Affinity DataKi: 2.67E+3nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 2.96E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 2.97E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 8.25E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 9.22E+3nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 1.42E+4nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataIC50: 0.00110nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataIC50: 0.00340nMAssay Description:Compound was tested for Adrenergic activity against Alpha-2 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataIC50: 0.0140nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataIC50: 0.0160nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair