TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.0600nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Binding affinity to muscarinic M3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Binding affinity to muscarinic M3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Binding affinity to muscarinic M3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.0900nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Binding affinity to muscarinic M3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.640nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.640nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 0.830nMAssay Description:Binding affinity to muscarinic M3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.850nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 1.02nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataKi: 1.51nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Rattus norvegicus (rat))
Pfizer
Pfizer
Affinity DataKi: 4nMAssay Description:PDE activity was monitored by measuring the hydrolysis of [3H]-cAMP to [3H]-AMP using a scintillation proximity assay (SPA). [3H]-AMP was captured by...More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of radiolabeled 4-(azetidin-1-yl)-3-[5-[4-(trifluoromethyl)phenyl]-1H-pyrazol-4-yl]-1-(tritritiomethyl)pyrazolo[3,4-d]pyrimidine from PD...More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Rattus norvegicus (rat))
Pfizer
Pfizer
Affinity DataKi: 12nMAssay Description:PDE activity was monitored by measuring the hydrolysis of [3H]-cAMP to [3H]-AMP using a scintillation proximity assay (SPA). [3H]-AMP was captured by...More data for this Ligand-Target Pair
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Rattus norvegicus (rat))
Pfizer
Pfizer
Affinity DataKi: 12nMAssay Description:PDE activity was monitored by measuring the hydrolysis of [3H]-cAMP to [3H]-AMP using a scintillation proximity assay (SPA). [3H]-AMP was captured by...More data for this Ligand-Target Pair
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Rattus norvegicus (rat))
Pfizer
Pfizer
Affinity DataKi: 12nMAssay Description:PDE activity was monitored by measuring the hydrolysis of [3H]-cAMP to [3H]-AMP using a scintillation proximity assay (SPA). [3H]-AMP was captured by...More data for this Ligand-Target Pair