TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Affinity DataIC50: 5nMAssay Description:Compound was evaluated for its inhibitory activity against the Caspase-9 enzymeMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 6.31nMAssay Description:Inhibition of human HRI kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Compound was evaluated for its inhibitory activity against the Caspase-7 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Compound was evaluated for its inhibitory activity against the Caspase-8 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of [3H]- DCKA binding to NMDA receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 7.94nMAssay Description:Inhibition of human HRI kinaseMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Oregon
Curated by ChEMBL
University Of Oregon
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of [3H]- DCKA binding to NMDA receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Oregon
Curated by ChEMBL
University Of Oregon
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Compound was evaluated for its inhibitory activity against the Caspase-6 enzymeMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 19.9nMAssay Description:Inhibition of human HRI kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Compound was evaluated for its inhibitory activity against the Caspase-1 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of [3H]- DCKA binding to NMDA receptor of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human recombinant Caspase-3 enzymeMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 31.6nMAssay Description:Inhibition of human HRI kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of [3H]- DCKA binding to NMDA receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Oregon
Curated by ChEMBL
University Of Oregon
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of [3H]- DCKA binding to NMDA receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Oregon
Curated by ChEMBL
University Of Oregon
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Oregon
Curated by ChEMBL
University Of Oregon
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 50.1nMAssay Description:Inhibition of human HRI kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibition of [3H]- DCKA binding to NMDA receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 63.1nMAssay Description:Inhibition of human HRI kinaseMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 63.1nMAssay Description:Inhibition of human HRI kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibitory activity against human recombinant Caspase-3 enzymeMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 79.4nMAssay Description:Inhibition of human HRI kinaseMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Oregon
Curated by ChEMBL
University Of Oregon
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against human recombinant Caspase-3 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against human recombinant Caspase-3 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against human recombinant Caspase-3 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Compound was evaluated for its inhibitory activity against the Calpain-1 enzymeMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of human HRI kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of [3H]- DCKA binding to NMDA receptor of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against human recombinant Caspase-3 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of [3H]- DCKA binding to NMDA receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Oregon
Curated by ChEMBL
University Of Oregon
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against human recombinant Caspase-3 enzymeMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Oregon
Curated by ChEMBL
University Of Oregon
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human HRI kinaseMore data for this Ligand-Target Pair