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Found 66 with Last Name = 'igarashi' and Initial = 'k'
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM50062599(3,5-Dimethyl-adamantan-1-ylamine | CHEMBL807 | EN3...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86155(TB-3-4)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86158(N1-n-octanesulfonyl-spermine)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86164(N1-DnsSpm | N1-dansyl-spermidine)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86157(Aminopropyl-cyclohexylamine | CAS_3312-60-5 | N-(3...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86153(CAS_180081 | MK-801 | NSC_180081)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86161(BE 4-4-4-4 | BE4444 | CAS_147510-59-6)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86165(Arcaine | CAS_2227 | CHEMBL102740 | NSC_2227)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM50038002(Benzamidine (Protonated) | CHEMBL20936 | CHEMBL537...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86166(DB-10)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86160(DB-3-3)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86162(DB-7)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86156(CAS_3037648 | MB-3 | NSC_3037648)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86163(CAS_9991 | MGBG | NSC_9991)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86164(N1-DnsSpm | N1-dansyl-spermidine)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM45440(4-[5-(4-amidinophenoxy)pentoxy]benzamidine;2-hydro...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM79403(3-aminopropyl-[4-(3-aminopropylamino)butyl]amine;h...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86154(Aminoguanidine | CAS_2146 | NSC_2146)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM76298(2-aminopropanoic acid [1-(4-chlorophenyl)-2-methyl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM85213(Agmatine | CAS_306-60-5 | CHEMBL58343 | NSC_199 | ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM72700(9-acridinamine;hydrate;hydrochloride | 9-aminoacri...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM86159(4-MB-3-3)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM50009371(1, 12-DB-3-4-3 | CHEMBL81614 | N,N'-Bis-(3-benzyla...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIonotropic glutamate receptor subunit Delta2(Xenopus)
State University of New York

Curated by PDSP Ki Database
LigandPNGBDBM50184779(4, 9-DB-3-4-3 | CHEMBL58084 | N,N'-Bis-(3-amino-pr...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50062599(3,5-Dimethyl-adamantan-1-ylamine | CHEMBL807 | EN3...)
Affinity DataIC50:  0.950nMAssay Description:Antagonist activity at recombinant GluN1/GluN2A receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as inhibition of glycine/gluta...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50492253(CHEMBL2398522)
Affinity DataIC50:  4.20nMAssay Description:Antagonist activity at recombinant GluN1/GluN2A receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as inhibition of glycine/gluta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50492252(CHEMBL55568)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at recombinant GluN1/GluN2A receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as inhibition of glycine/gluta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476423(CHEMBL228435)
Affinity DataIC50:  72nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476427(CHEMBL228436)
Affinity DataIC50:  78nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476433(CHEMBL228486)
Affinity DataIC50:  83nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50492255(CHEMBL2009741)
Affinity DataIC50:  89nMAssay Description:Antagonist activity at recombinant GluN1/GluN2A receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as inhibition of glycine/gluta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476427(CHEMBL228436)
Affinity DataIC50:  108nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476432(CHEMBL228437)
Affinity DataIC50:  108nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476430(CHEMBL388315)
Affinity DataIC50:  111nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476424(CHEMBL228380)
Affinity DataIC50:  117nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476432(CHEMBL228437)
Affinity DataIC50:  127nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataIC50:  138nMAssay Description:Antagonist activity at recombinant GluN1/GluN2A receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as inhibition of glycine/gluta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476423(CHEMBL228435)
Affinity DataIC50:  142nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476433(CHEMBL228486)
Affinity DataIC50:  145nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476430(CHEMBL388315)
Affinity DataIC50:  166nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476431(CHEMBL390521)
Affinity DataIC50:  189nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476425(CHEMBL228325)
Affinity DataIC50:  198nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476422(CHEMBL390304)
Affinity DataIC50:  199nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476422(CHEMBL390304)
Affinity DataIC50:  203nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476431(CHEMBL390521)
Affinity DataIC50:  211nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476426(CHEMBL390305)
Affinity DataIC50:  215nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476421(CHEMBL228378)
Affinity DataIC50:  240nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50492256(CHEMBL2398521)
Affinity DataIC50:  257nMAssay Description:Antagonist activity at recombinant GluN1/GluN2A receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as inhibition of glycine/gluta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476424(CHEMBL228380)
Affinity DataIC50:  270nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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