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Found 38 with Last Name = 'igari' and Initial = 'n'
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030174((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030199((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  1.70nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030178((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  1.70nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030204((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  1.80nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030210((R)-1-[1-(2-Dimethylamino-ethyl)-1H-indole-3-carbo...)
Affinity DataIC50:  3.5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030181((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  3.5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030182((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  3.5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030188((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  4.30nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50407171(CHEMBL2114031)
Affinity DataIC50:  4.60nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030179((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  4.90nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030180((R)-4-Hydroxy-1-(1H-indazole-3-carbonyl)-pyrrolidi...)
Affinity DataIC50:  5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030203(1-(1H-Indole-3-carbonyl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50:  5.40nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030177((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  5.40nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030197((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  6.40nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030185((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  7nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50407172(CHEMBL2115107)
Affinity DataIC50:  7.40nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030192((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  7.60nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030189(1-(1H-Indole-3-carbonyl)-azetidine-2-carboxylic ac...)
Affinity DataIC50:  8nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030176(CHEMBL65703 | N*1*-[(R)-1-(Benzyl-methyl-carbamoyl...)
Affinity DataIC50:  9nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030187((R)-4-Hydroxy-1-[(E)-(3-phenyl-acryloyl)]-pyrrolid...)
Affinity DataIC50:  9nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030205((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  9.20nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030191((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  10nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030190(1H-Indole-3-carboxylic acid {1-[(R)-1-(benzyl-meth...)
Affinity DataIC50:  11nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030194((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  12nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030184((R)-4-Hydroxy-1-(3-phenyl-propionyl)-pyrrolidine-2...)
Affinity DataIC50:  14nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030186(1H-Indole-3-carboxylic acid {5-amino-1-[(R)-1-(ben...)
Affinity DataIC50:  14nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030208((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  14nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030209((R)-4-Hydroxy-1-(1-isopropyl-1H-indole-3-carbonyl)...)
Affinity DataIC50:  16nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030198((R)-1-(Benzo[b]thiophene-2-carbonyl)-4-hydroxy-pyr...)
Affinity DataIC50:  20nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030175((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  23nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030207(1H-Indole-3-carboxylic acid {1-[(R)-1-(benzyl-meth...)
Affinity DataIC50:  23nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030202((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  25nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030206((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  27nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030201((R)-4-Hydroxy-1-(4-phenyl-butyryl)-pyrrolidine-2-c...)
Affinity DataIC50:  32nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030195(1H-Indole-3-carboxylic acid {[(R)-1-(benzyl-methyl...)
Affinity DataIC50:  33nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030193((3-{(R)-2-[(R)-1-(Benzyl-methyl-carbamoyl)-2-pheny...)
Affinity DataIC50:  50nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030200((R)-4-Hydroxy-1-phenylacetyl-pyrrolidine-2-carboxy...)
Affinity DataIC50:  139nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50030183(5-Hydroxy-1-(1H-indole-3-carbonyl)-piperidine-2-ca...)
Affinity DataIC50:  289nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed