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Found 113 with Last Name = 'ingalls' and Initial = 'cl'
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50161957(4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(p...)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50161957(4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(p...)
Affinity DataIC50:  0.180nMAssay Description:Inhibition of human EGFR in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM31090((E)-N-[4-(3-chloro-4-fluoro-anilino)-3-cyano-7-eth...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM3032(CHEMBL1204168 | CHEMBL29197 | N-(3-bromophenyl)-6,...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209886((2E)-4-(dimethylamino)-N-[7-ethoxy-4-({4-[(3-fluor...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152049(3-(2,4-Dichloro-phenyl)-7-dicyclopropylmethyl-8-et...)
Affinity DataIC50:  6nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152033(7-(1-Cyclopropyl-butyl)-3-(2,4-dichloro-phenyl)-8-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209878((2E)-N-[4-({4-[(3-chlorobenzyl)oxy]-3,6-dioxocyclo...)
Affinity DataIC50:  12.2nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152054(7-(1-Cyclopropyl-propyl)-3-(2,4-dichloro-phenyl)-8...)
Affinity DataIC50:  14nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152059(3-(2,4-Dichloro-phenyl)-8-ethyl-7-(1-ethyl-pentyl)...)
Affinity DataIC50:  18nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209879((2E)-N-(4-{[4-(benzyloxy)-3,6-dioxocyclohexa-1,4-d...)
Affinity DataIC50:  18.7nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152043(8-Ethyl-1-methyl-7-(1-propyl-butyl)-3-(2,4,6-trime...)
Affinity DataIC50:  22nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209883((2E)-4-(dimethylamino)-N-[7-ethoxy-4-({4-[(3-methy...)
Affinity DataIC50:  24.9nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152031(7-(1-Cyclobutyl-ethyl)-3-(2,4-dichloro-phenyl)-8-e...)
Affinity DataIC50:  26nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152055(3-(2-Chloro-4-methoxy-phenyl)-8-ethyl-1-methyl-7-(...)
Affinity DataIC50:  27nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  27.3nMAssay Description:Inhibition of human VEGFR2 in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM31090((E)-N-[4-(3-chloro-4-fluoro-anilino)-3-cyano-7-eth...)
Affinity DataIC50:  34.9nMAssay Description:Inhibition of human EGFR in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209878((2E)-N-[4-({4-[(3-chlorobenzyl)oxy]-3,6-dioxocyclo...)
Affinity DataIC50:  35.6nMAssay Description:Inhibition of human EGFR in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152044(3-(2,4-Dichloro-phenyl)-8-ethyl-7-(1-methoxymethyl...)
Affinity DataIC50:  43nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209886((2E)-4-(dimethylamino)-N-[7-ethoxy-4-({4-[(3-fluor...)
Affinity DataIC50:  43.1nMAssay Description:Inhibition of human EGFR in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209877(2-(3-fluorobenzyloxy)-5-(6-methoxy-7-(2-methoxyeth...)
Affinity DataIC50:  46.1nMAssay Description:Inhibition of human VEGFR2 in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209884((2E)-4-(dimethylamino)-N-(4-{[3,6-dioxo-4-(2-thien...)
Affinity DataIC50:  47.5nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152030(3-(2-Chloro-4-isopropyl-phenyl)-8-ethyl-1-methyl-7...)
Affinity DataIC50:  50nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209882(2-(3-methoxybenzyloxy)-5-(6-methoxy-7-(2-methoxyet...)
Affinity DataIC50:  50.2nMAssay Description:Inhibition of human VEGFR2 in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152035(3-(2,4-Dichloro-phenyl)-8-ethyl-7-(1-ethyl-2-methy...)
Affinity DataIC50:  51nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152037(3-(2,4-Dichloro-phenyl)-8-ethyl-1-methyl-7-(1-meth...)
Affinity DataIC50:  52nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209888(2-(benzyloxy)-5-(6-methoxy-7-(2-methoxyethoxy)quin...)
Affinity DataIC50:  53.7nMAssay Description:Inhibition of human VEGFR2 in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152038(3-(2,4-Dichloro-phenyl)-8-ethyl-1-methyl-7-(1-prop...)
Affinity DataIC50:  54nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152056(7-(1-Cyclopropyl-ethyl)-3-(2,4-dichloro-phenyl)-8-...)
Affinity DataIC50:  55nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152053(3-(2,4-Dichloro-phenyl)-8-ethyl-1-methyl-7-(1-prop...)
Affinity DataIC50:  75nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209884((2E)-4-(dimethylamino)-N-(4-{[3,6-dioxo-4-(2-thien...)
Affinity DataIC50:  76.2nMAssay Description:Inhibition of human VEGFR2 in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209878((2E)-N-[4-({4-[(3-chlorobenzyl)oxy]-3,6-dioxocyclo...)
Affinity DataIC50:  80.2nMAssay Description:Inhibition of human VEGFR2 in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209885((2E)-4-(dimethylamino)-N-(4-{[3,6-dioxo-4-(pyridin...)
Affinity DataIC50:  90.8nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM3032(CHEMBL1204168 | CHEMBL29197 | N-(3-bromophenyl)-6,...)
Affinity DataIC50: >100nMAssay Description:Inhibition of human EGFR in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209879((2E)-N-(4-{[4-(benzyloxy)-3,6-dioxocyclohexa-1,4-d...)
Affinity DataIC50:  102nMAssay Description:Inhibition of human VEGFR2 in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209875((2E)-4-(dimethylamino)-N-[7-ethoxy-4-({4-[(3-metho...)
Affinity DataIC50:  107nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209881((2E)-4-(dimethylamino)-N-[7-ethoxy-4-({4-[2-fluoro...)
Affinity DataIC50:  109nMAssay Description:Inhibition of human VEGFR2 in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209880((2E)-N-[4-({4-[(3,4-difluorobenzyl)oxy]-3,6-dioxoc...)
Affinity DataIC50:  112nMAssay Description:Inhibition of human VEGFR2 in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152034(3-(2,4-Dichloro-phenyl)-8-ethyl-7-(1-ethyl-propyl)...)
Affinity DataIC50:  112nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  112nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152040(3-(2-Chloro-4-methoxy-phenyl)-7-(1-cyclopropyl-pro...)
Affinity DataIC50:  113nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209886((2E)-4-(dimethylamino)-N-[7-ethoxy-4-({4-[(3-fluor...)
Affinity DataIC50:  113nMAssay Description:Inhibition of human VEGFR2 in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209885((2E)-4-(dimethylamino)-N-(4-{[3,6-dioxo-4-(pyridin...)
Affinity DataIC50:  135nMAssay Description:Inhibition of human VEGFR2 in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209888(2-(benzyloxy)-5-(6-methoxy-7-(2-methoxyethoxy)quin...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human VEGFR2 in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152051(8-Ethyl-3-(4-methoxy-2-pyridin-3-ylmethyl-phenyl)-...)
Affinity DataIC50:  161nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209880((2E)-N-[4-({4-[(3,4-difluorobenzyl)oxy]-3,6-dioxoc...)
Affinity DataIC50:  167nMAssay Description:Inhibition of human EGFR in presence of 1 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152061(3-(4-Chloro-phenyl)-8-ethyl-1-methyl-7-(1-propyl-b...)
Affinity DataIC50:  173nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209883((2E)-4-(dimethylamino)-N-[7-ethoxy-4-({4-[(3-methy...)
Affinity DataIC50:  173nMAssay Description:Inhibition of human EGFR in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50209878((2E)-N-[4-({4-[(3-chlorobenzyl)oxy]-3,6-dioxocyclo...)
Affinity DataIC50:  179nMAssay Description:Inhibition of human VEGFR2 in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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