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Found 2730 with Last Name = 'ito' and Initial = 'r'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057433(CHEMBL278806 | [2-(5-Fluoro-chroman-8-yloxy)-ethyl...)
Affinity DataKi:  0.0500nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057432(CHEMBL25215 | [2-(Chroman-8-yloxy)-ethyl]-[4-(4-me...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065562(CHEMBL96279 | [2-(6-Fluoro-2,2-dimethyl-chroman-8-...)
Affinity DataKi:  0.149nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065578(CHEMBL419147 | [2-(6-Fluoro-2H-chromen-8-yloxy)-et...)
Affinity DataKi:  0.159nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065555(CHEMBL96578 | [2-(6-Fluoro-2-methyl-chroman-8-ylox...)
Affinity DataKi:  0.188nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85052(BIM 23197 | BIM-23197)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057436(CHEMBL25213 | [2-(6-Fluoro-chroman-8-yloxy)-ethyl]...)
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM18860((2R)-2-amino-3-[4-(4-hydroxy-3-iodophenoxy)-3,5-di...)
Affinity DataKi:  0.220nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor alpha (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057436(CHEMBL25213 | [2-(6-Fluoro-chroman-8-yloxy)-ethyl]...)
Affinity DataKi:  0.221nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057436(CHEMBL25213 | [2-(6-Fluoro-chroman-8-yloxy)-ethyl]...)
Affinity DataKi:  0.259nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057436(CHEMBL25213 | [2-(6-Fluoro-chroman-8-yloxy)-ethyl]...)
Affinity DataKi:  0.260nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065573(CHEMBL96222 | [2-(6-Fluoro-2-methyl-chroman-8-ylox...)
Affinity DataKi:  0.270nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057434(8-{2-[4-(4-Methoxy-phenyl)-butylamino]-ethoxy}-chr...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065578(CHEMBL419147 | [2-(6-Fluoro-2H-chromen-8-yloxy)-et...)
Affinity DataKi:  0.288nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065573(CHEMBL96222 | [2-(6-Fluoro-2-methyl-chroman-8-ylox...)
Affinity DataKi:  0.312nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50370683(CHEMBL1169543)
Affinity DataKi:  0.320nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85051(BIM-23190)
Affinity DataKi:  0.340nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057429(CHEMBL22328 | [2-(7-Fluoro-chroman-8-yloxy)-ethyl]...)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50063839(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM18869(2-{3,5-dichloro-4-[4-hydroxy-3-(propan-2-yl)phenox...)
Affinity DataKi:  0.370nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor beta (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM82465(BIM 23023 | BIM-23023 | D-Phe-L-Cys(1)-L-Tyr-D-Trp...)
Affinity DataKi:  0.420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065562(CHEMBL96279 | [2-(6-Fluoro-2,2-dimethyl-chroman-8-...)
Affinity DataKi:  0.435nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057428(CHEMBL22682 | [2-(6-Chloro-chroman-8-yloxy)-ethyl]...)
Affinity DataKi:  0.490nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM18860((2R)-2-amino-3-[4-(4-hydroxy-3-iodophenoxy)-3,5-di...)
Affinity DataKi:  0.550nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor beta (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057432(CHEMBL25215 | [2-(Chroman-8-yloxy)-ethyl]-[4-(4-me...)
Affinity DataKi:  0.580nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity of the compound was evaluated against Dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand; ND = Not determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065563(6-Fluoro-8-{2-[4-(4-methoxy-phenyl)-butylamino]-et...)
Affinity DataKi:  0.724nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065563(6-Fluoro-8-{2-[4-(4-methoxy-phenyl)-butylamino]-et...)
Affinity DataKi:  0.724nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  0.75nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057431(CHEMBL21475 | [4-(4-Methoxy-phenyl)-butyl]-[2-(6-m...)
Affinity DataKi:  0.780nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50258672(CHEMBL513681 | [4-(2,3,4,5-Tetrahydro-1,3-dimethyl...)
Affinity DataKi:  0.794nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50370683(CHEMBL1169543)
Affinity DataKi:  0.820nMAssay Description:Binding affinity for rat salivary gland muscarinic acetylcholine receptor M3 using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  0.880nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50175574((S)-1-Thiophen-3-yl-3,4-dihydro-1H-isoquinoline-2-...)
Affinity DataKi:  0.950nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50282641(CHEMBL4160732)
Affinity DataKi:  1nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin receptor 1(Homo sapiens (Human))
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563230(CHEMBL4754949)
Affinity DataKi:  1.10nMAssay Description:Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM82253(BIM 23052 | CAS_133073-82-2)
Affinity DataKi:  1.22nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50282638(CHEMBL4175851)
Affinity DataKi:  1.30nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057428(CHEMBL22682 | [2-(6-Chloro-chroman-8-yloxy)-ethyl]...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50175570((S)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxy...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  1.43nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50175581(Benzhydryl-carbamic acid 1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  1.77nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057434(8-{2-[4-(4-Methoxy-phenyl)-butylamino]-ethoxy}-chr...)
Affinity DataKi:  1.80nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057431(CHEMBL21475 | [4-(4-Methoxy-phenyl)-butyl]-[2-(6-m...)
Affinity DataKi:  1.80nMAssay Description:In vitro radioligand binding assay on Dopamine receptor D2 of rat striatum using [3H]- spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50175575(1-Thiophen-2-yl-3,4-dihydro-1H-isoquinoline-2-carb...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50175575(1-Thiophen-2-yl-3,4-dihydro-1H-isoquinoline-2-carb...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50282631(CHEMBL4175454)
Affinity DataKi:  1.80nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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