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Found 869 with Last Name = 'jain' and Initial = 'a'
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034332((3aS,9bS)-3-Propyl-2,3,3a,4,5,9b-hexahydro-1H-benz...)
Affinity DataKi:  0.100nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034322((3aS,9bS)-3-Allyl-9-methoxy-2,3,3a,4,5,9b-hexahydr...)
Affinity DataKi:  0.200nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034331((3aS,9bS)-9-Methoxy-3-propyl-2,3,3a,4,5,9b-hexahyd...)
Affinity DataKi:  0.200nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'/beta(Homo sapiens (Human))
Cylene Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataKi:  0.220nMAssay Description:Inhibition of human recombinant CK2alpha/CK2beta using RRRDDDSDDD peptide as substrate by radiometric assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034348((2aR,8bR)-2-Allyl-1,2,2a,3,4,8b-hexahydro-naphtho[...)
Affinity DataKi:  0.300nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034360((3aR,9bS)-3-Allyl-2,3,3a,4,5,9b-hexahydro-1H-benzo...)
Affinity DataKi:  0.300nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034333((2S,3aR,9bS)-2-Methyl-3-propyl-2,3,3a,4,5,9b-hexah...)
Affinity DataKi:  1nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034362((R)-6-Dipropylamino-1,2,6,7-tetrahydro-5H-pyrido[3...)
Affinity DataKi:  2.20nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034342((3aR,9bS) 3-Propyl-2,3,3a,4,5,9b-hexahydro-1H-benz...)
Affinity DataKi:  3nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(MOUSE)
National Institute Of Pharmaceutical Education And Research (Niper) - Ahmedabad

Curated by ChEMBL
LigandPNGBDBM50591643(CHEMBL5172956)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to mouse PKC-alpha assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034339((3aR,9bR)-3-Allyl-9-methoxy-2,3,3a,4,5,9b-hexahydr...)
Affinity DataKi:  4.70nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034321((3aR,9bR)-3-Allyl-2,3,3a,4,5,9b-hexahydro-1H-benzo...)
Affinity DataKi:  4.90nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384714(CHEMBL2037200)
Affinity DataKi:  5nMAssay Description:Reversible inhibition of human recombinant Pim1 using RSRHSSYPAGT as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034357((2aR,8bR)-2-Allyl-8-methoxy-1,2,2a,3,4,8b-hexahydr...)
Affinity DataKi:  5.90nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(MOUSE)
National Institute Of Pharmaceutical Education And Research (Niper) - Ahmedabad

Curated by ChEMBL
LigandPNGBDBM50591642(CHEMBL5205471)
Affinity DataKi:  8.70nMAssay Description:Binding affinity to mouse PKC-alpha assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034323((2 beta-methyl) 8-Methoxy-2-methyl-1-propyl-2,3,3a...)
Affinity DataKi:  11nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034335((3aR,9bR)-3-Allyl-2,3,3a,4,5,9b-hexahydro-1H-benzo...)
Affinity DataKi:  11nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50383265(CHEMBL2032368)
Affinity DataKi:  11nMAssay Description:Inhibition of human Pim-1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate preincubated for 15 mins prior substrate addition measured after 45 mins by fluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034356((3aR,9bR)-3-Allyl-2,3,3a,4,5,9b-hexahydro-1H-benzo...)
Affinity DataKi:  16nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034329((2R,3aR,9bS)-2-Methyl-3-propyl-2,3,3a,4,5,9b-hexah...)
Affinity DataKi:  16nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034364((3aR,9bR)-3-Allyl-6-methoxy-2,3,3a,4,5,9b-hexahydr...)
Affinity DataKi:  16nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034324((3aS,9aR) 5-Methoxy-1-propyl-2,3,3a,4,9,9a-hexahyd...)
Affinity DataKi:  17nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034354((R)-5-Dipropylamino-5,6-dihydro-1H,4H-imidazo[4,5,...)
Affinity DataKi:  24.8nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034347((3aS,9aR)-1-(cyclopropylmethyl)-5-methoxy-2,3,3a,4...)
Affinity DataKi:  29nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034312((3aS,9aR)-5-Methoxy-2,3,3a,4,9,9a-hexahydro-1H-ben...)
Affinity DataKi:  29nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034337((3aR,9bS)-3-Allyl-2,3,3a,4,5,9b-hexahydro-1H-benzo...)
Affinity DataKi:  31nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034352((3aS,9aR) 1-Propyl-2,3,3a,4,9,9a-hexahydro-1H-benz...)
Affinity DataKi:  36nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034358((3aR,9bS)-3-Propyl-2,3,3a,4,5,9b-hexahydro-1H-benz...)
Affinity DataKi:  37nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034350((3aS,9aR) 1-Allyl-5-methoxy-2,3,3a,4,9,9a-hexahydr...)
Affinity DataKi:  41nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034316((3aR,9bR)-3-Propyl-2,3,3a,4,5,9b-hexahydro-1H-benz...)
Affinity DataKi:  44nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034330((3aR,9bS) 3-Allyl-9-methoxy-2,3,3a,4,5,9b-hexahydr...)
Affinity DataKi:  49nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034359((3aS,9bS)-3-Allyl-2,3,3a,4,5,9b-hexahydro-1H-benzo...)
Affinity DataKi:  54nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034346((3aS,9aR) 1-Allyl-2,3,3a,4,9,9a-hexahydro-1H-benzo...)
Affinity DataKi:  56nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034336((3aR,9bR)-3-Cyclopropylmethyl-6-methoxy-2,3,3a,4,5...)
Affinity DataKi:  66nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034326((3aR,9bR)-6-Methoxy-3-propyl-2,3,3a,4,5,9b-hexahyd...)
Affinity DataKi:  66nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034338((3aS,9aR)-1-Cyclopropylmethyl-2,3,3a,4,9,9a-hexahy...)
Affinity DataKi:  69nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034353((3aS,9aR)-1-Allyl-8-methoxy-2,3,3a,4,9,9a-hexahydr...)
Affinity DataKi:  104nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034361((3aS,9aR)-1-Benzyl-5-methoxy-2,3,3a,4,9,9a-hexahyd...)
Affinity DataKi:  127nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034344((3aS,9aS)-1-Allyl-8-methoxy-2,3,3a,4,9,9a-hexahydr...)
Affinity DataKi:  145nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034327((3aR,9bS) 9-Methoxy-3-propyl-2,3,3a,4,5,9b-hexahyd...)
Affinity DataKi:  186nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034317((3aS,9bS)-3-Allyl-6-methoxy-2,3,3a,4,5,9b-hexahydr...)
Affinity DataKi:  236nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034340((3aR,9bS)-9-Methoxy-3-phenethyl-2,3,3a,4,5,9b-hexa...)
Affinity DataKi:  317nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034341((3aR,9bS)-3-allyl-6-methoxy-2,3,3a,4,5,9b-hexahydr...)
Affinity DataKi:  333nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034349((3aR,9bR)-3-Propyl-2,3,3a,4,5,9b-hexahydro-1H-benz...)
Affinity DataKi:  338nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034325((2 alpha-methyl) 8-Methoxy-2-methyl-1-propyl-2,3,3...)
Affinity DataKi:  384nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034328((3aS,9bS)-9-Methoxy-3-phenethyl-2,3,3a,4,5,9b-hexa...)
Affinity DataKi:  442nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034334((3aR,9aR)-1-Allyl-2,3,3a,4,9,9a-hexahydro-1H-benzo...)
Affinity DataKi:  470nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034310((3aR,9aR)-1-Propyl-2,3,3a,4,9,9a-hexahydro-1H-benz...)
Affinity DataKi:  470nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034343((3aS,9aS)-1-Cyclopropylmethyl-5-methoxy-2,3,3a,4,9...)
Affinity DataKi:  721nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034319((3aS,9aS)-1-Propyl-2,3,3a,4,9,9a-hexahydro-1H-benz...)
Affinity DataKi:  1.00E+3nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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