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maximum 50k data
Found 37 with Last Name = 'jin' and Initial = 'lw'
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476303(CHEMBL227521)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476296(CHEMBL228033)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476855(CHEMBL232112)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476293(CHEMBL227495)
Affinity DataKi:  1.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476287(CHEMBL224096)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476298(CHEMBL223285)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476299(CHEMBL228034)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476292(CHEMBL227577)
Affinity DataKi:  3.10nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476301(CHEMBL413436)
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476300(CHEMBL389671)
Affinity DataKi:  3.80nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476291(CHEMBL227674)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476297(CHEMBL227576)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476850(CHEMBL232114)
Affinity DataKi:  6.20nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476852(CHEMBL231917)
Affinity DataKi:  6.70nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476848(CHEMBL231916)
Affinity DataKi:  9.20nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476853(CHEMBL398059)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476288(CHEMBL373663)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476854(CHEMBL232113)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476851(CHEMBL231918)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476849(CHEMBL231915)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476302(CHEMBL227751)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476286(CHEMBL226610)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476294(CHEMBL227752)
Affinity DataKi:  68nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476290(CHEMBL227625)
Affinity DataKi:  76nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476295(CHEMBL373548)
Affinity DataKi:  106nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476289(CHEBI:51579 | DIPHENYLACETYLENE)
Affinity DataKi:  175nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kansas State University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  33nMAssay Description:Inhibition of GSK3beta (unknown origin) assessed as luminescence intensity by luminometryMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50046523(CHEMBL495039)
Affinity DataIC50:  35nMAssay Description:Inhibition of GSK3beta (unknown origin) assessed as luminescence intensity by luminometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50005944(2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)
Affinity DataIC50:  200nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50397451(CHEMBL2170736)
Affinity DataIC50:  300nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50397448(CHEMBL2170728)
Affinity DataIC50:  800nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50397452(CHEMBL520938)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50397450(CHEMBL2170821)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50397449(CHEMBL2170832)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50046524(CHEMBL3311235)
Affinity DataIC50:  2.40E+5nMAssay Description:Inhibition of GSK3beta (unknown origin) assessed as luminescence intensity by luminometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50046525(CHEMBL3311239)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of GSK3beta (unknown origin) assessed as luminescence intensity by luminometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50046526(CHEMBL3311242)
Affinity DataIC50:  7.50E+5nMAssay Description:Inhibition of GSK3beta (unknown origin) assessed as luminescence intensity by luminometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed