TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 6.70nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 9.20nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 76nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 106nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 175nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of GSK3beta (unknown origin) assessed as luminescence intensity by luminometryMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of GSK3beta (unknown origin) assessed as luminescence intensity by luminometryMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibition of GSK3beta (unknown origin) assessed as luminescence intensity by luminometryMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of GSK3beta (unknown origin) assessed as luminescence intensity by luminometryMore data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+5nMAssay Description:Inhibition of GSK3beta (unknown origin) assessed as luminescence intensity by luminometryMore data for this Ligand-Target Pair