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Found 561 with Last Name = 'jones' and Initial = 'tr'
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50405732(CHEMBL290277)
Affinity DataKi:  0.0410nMAssay Description:Compound was tested for inhibition of human (WI-L2) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50405733(CHEMBL406575)
Affinity DataKi:  0.0420nMAssay Description:Compound was tested for inhibition of human (WI-L2) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50405731(CHEMBL295708)
Affinity DataKi:  0.0720nMAssay Description:Compound was tested for inhibition of human (WI-L2) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50405730(CHEMBL295681)
Affinity DataKi:  0.224nMAssay Description:Compound was tested for inhibition of human (WI-L2) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Rattus norvegicus (rat))
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50006906(2-{4-[(2-Amino-4-hydroxy-quinazolin-6-ylmethyl)-am...)
Affinity DataKi:  0.580nMAssay Description:Compound was evaluated for the inhibition of partially purified rat liver Dihydrofolate reductase (DHFR) enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM18771((2S)-2-[(4-{[(2-amino-4-oxo-1,4-dihydroquinazolin-...)
Affinity DataKi:  3.40nMAssay Description:Binding affinity against Thymidylate synthase was measured in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Rattus norvegicus (rat))
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50017876(2-{4-[(2-Amino-4-oxo-3,4-dihydro-quinazolin-6-ylme...)
Affinity DataKi:  3.90nMAssay Description:Compound was evaluated for the inhibition of partially purified rat liver Dihydrofolate reductase (DHFR) enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50008294(2-(4-(((2-amino-4-oxo-1,4-dihydroquinazolin-6-yl)m...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity was evaluated against thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50027900(2-{4-[(2-Amino-4-oxo-3,4-dihydro-quinazolin-6-ylme...)
Affinity DataKi:  7nMAssay Description:Compound was tested for inhibition of human (WI-L2) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50006687((S)-2-(4-(((2-methyl-4-oxo-3,4-dihydroquinazolin-6...)
Affinity DataKi:  10nMAssay Description:Binding affinity against Thymidylate synthase was measured in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Rattus norvegicus (rat))
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50006907(2-{4-[(4-Oxo-3,4-dihydro-quinazolin-6-ylmethyl)-am...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for the inhibition of partially purified rat liver Dihydrofolate reductase (DHFR) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50011244(6-{[(4-Benzenesulfonyl-phenyl)-prop-2-ynyl-amino]-...)
Affinity DataKi:  12nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50011244(6-{[(4-Benzenesulfonyl-phenyl)-prop-2-ynyl-amino]-...)
Affinity DataKi:  12nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50008294(2-(4-(((2-amino-4-oxo-1,4-dihydroquinazolin-6-yl)m...)
Affinity DataKi:  14nMAssay Description:Binding affinity was evaluated against dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056521(6-{[(4-Benzenesulfonyl-3-fluoro-phenyl)-prop-2-yny...)
Affinity DataKi:  20nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056516(6-({[4-(2-Chloro-benzenesulfonyl)-phenyl]-prop-2-y...)
Affinity DataKi:  21nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056519(6-{[(4-Benzenesulfonyl-3-chloro-phenyl)-prop-2-yny...)
Affinity DataKi:  24nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50011244(6-{[(4-Benzenesulfonyl-phenyl)-prop-2-ynyl-amino]-...)
Affinity DataKi:  25nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056520(2-Methyl-6-({prop-2-ynyl-[4-(toluene-2-sulfonyl)-p...)
Affinity DataKi:  26nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056518(6-{[(4-Benzenesulfinyl-3-chloro-phenyl)-prop-2-yny...)
Affinity DataKi:  27nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056518(6-{[(4-Benzenesulfinyl-3-chloro-phenyl)-prop-2-yny...)
Affinity DataKi:  27nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50014480((S)-2-(4-(((4-oxo-3,4-dihydroquinazolin-6-yl)methy...)
Affinity DataKi:  27nMAssay Description:Concentration required for in vitro inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056519(6-{[(4-Benzenesulfonyl-3-chloro-phenyl)-prop-2-yny...)
Affinity DataKi:  33nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056516(6-({[4-(2-Chloro-benzenesulfonyl)-phenyl]-prop-2-y...)
Affinity DataKi:  33nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056519(6-{[(4-Benzenesulfonyl-3-chloro-phenyl)-prop-2-yny...)
Affinity DataKi:  33nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056516(6-({[4-(2-Chloro-benzenesulfonyl)-phenyl]-prop-2-y...)
Affinity DataKi:  33nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50012245(6-{[(4-Benzenesulfonyl-3-trifluoromethyl-phenyl)-p...)
Affinity DataKi:  37nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056521(6-{[(4-Benzenesulfonyl-3-fluoro-phenyl)-prop-2-yny...)
Affinity DataKi:  43nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056521(6-{[(4-Benzenesulfonyl-3-fluoro-phenyl)-prop-2-yny...)
Affinity DataKi:  43nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056523(2-Methyl-6-({prop-2-ynyl-[4-(toluene-2-sulfinyl)-p...)
Affinity DataKi:  45nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056523(2-Methyl-6-({prop-2-ynyl-[4-(toluene-2-sulfinyl)-p...)
Affinity DataKi:  45nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056515(6-({[4-(2-Chloro-benzenesulfinyl)-phenyl]-prop-2-y...)
Affinity DataKi:  46nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056515(6-({[4-(2-Chloro-benzenesulfinyl)-phenyl]-prop-2-y...)
Affinity DataKi:  46nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50012245(6-{[(4-Benzenesulfonyl-3-trifluoromethyl-phenyl)-p...)
Affinity DataKi:  50nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056514(6-{[(4-Benzenesulfinyl-3-fluoro-phenyl)-prop-2-yny...)
Affinity DataKi:  50nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056518(6-{[(4-Benzenesulfinyl-3-chloro-phenyl)-prop-2-yny...)
Affinity DataKi:  54nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056520(2-Methyl-6-({prop-2-ynyl-[4-(toluene-2-sulfonyl)-p...)
Affinity DataKi:  56nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056520(2-Methyl-6-({prop-2-ynyl-[4-(toluene-2-sulfonyl)-p...)
Affinity DataKi:  56nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Rattus norvegicus (rat))
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50017875(2-{4-[Ethyl-(4-oxo-3,4-dihydro-quinazolin-6-ylmeth...)
Affinity DataKi:  58nMAssay Description:Compound was evaluated for the inhibition of partially purified rat liver Dihydrofolate reductase (DHFR) enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50049941(6-{[(4-Benzenesulfinyl-phenyl)-prop-2-ynyl-amino]-...)
Affinity DataKi:  61nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056522(6-{[(4-Benzenesulfinyl-3-trifluoromethyl-phenyl)-p...)
Affinity DataKi:  70nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056522(6-{[(4-Benzenesulfinyl-3-trifluoromethyl-phenyl)-p...)
Affinity DataKi:  70nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Rattus norvegicus (rat))
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50008294(2-(4-(((2-amino-4-oxo-1,4-dihydroquinazolin-6-yl)m...)
Affinity DataKi:  75nMAssay Description:Compound was evaluated for the inhibition of partially purified rat liver Dihydrofolate reductase(DHFR) enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Rattus norvegicus (rat))
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM18771((2S)-2-[(4-{[(2-amino-4-oxo-1,4-dihydroquinazolin-...)
Affinity DataKi:  75nMAssay Description:Inhibitory activity against Dihydrofolate reductase in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056514(6-{[(4-Benzenesulfinyl-3-fluoro-phenyl)-prop-2-yny...)
Affinity DataKi:  88nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056514(6-{[(4-Benzenesulfinyl-3-fluoro-phenyl)-prop-2-yny...)
Affinity DataKi:  88nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056522(6-{[(4-Benzenesulfinyl-3-trifluoromethyl-phenyl)-p...)
Affinity DataKi:  110nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056517(2-Methyl-6-({prop-2-ynyl-[4-(toluene-2-sulfonyl)-3...)
Affinity DataKi:  150nMAssay Description:Binding affinity against recombinant human thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056517(2-Methyl-6-({prop-2-ynyl-[4-(toluene-2-sulfonyl)-3...)
Affinity DataKi:  160nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Pedagogical University

Curated by ChEMBL
LigandPNGBDBM50056517(2-Methyl-6-({prop-2-ynyl-[4-(toluene-2-sulfonyl)-3...)
Affinity DataKi:  160nMAssay Description:Binding affinity against recombinant thymidylate synthase in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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