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Found 105 with Last Name = 'käck' and Initial = 'h'
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50339997((R)-2-(3-amino-1-phenylpropoxy)-4-chlorobenzonitri...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant iNOSMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50339998((R)-2-(3-amino-1-phenylpropylthio)-4-chlorobenzoni...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50340003((R)-2-(3-amino-1-phenylpropylthio)-6-methylnicotin...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50340004((R)-2-(3-amino-1-(isoxazol-5-yl)propoxy)-6-(triflu...)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of human recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50340002(2-[[(1R)-3-Amino-1-phenylpropyl]oxy]-4-chloro-5-fl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50339996((R)-4-chloro-2-(3-(methylamino)-1-phenylpropoxy)be...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421064(CHEMBL2087855)
Affinity DataIC50:  13nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50339995((R)-3-(2,5-dichlorophenoxy)-N-methyl-3-phenylpropa...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421055(CHEMBL1652588)
Affinity DataIC50:  24nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50215445(5-(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropy...)
Affinity DataIC50:  25nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421065(CHEMBL2087856)
Affinity DataIC50:  28nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50262114(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropylme...)
Affinity DataIC50:  34nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421042(CHEMBL2087619)
Affinity DataIC50:  39nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50124535(1-(6-CYANO-3-PYRIDYLCARBONYL)-5',8'-DIFLUOROSPIRO[...)
Affinity DataIC50:  41nMAssay Description:Inhibition of human recombinant iNOSMore data for this Ligand-Target Pair
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421086(CHEMBL2087620)
Affinity DataIC50:  41nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421066(CHEMBL2087857)
Affinity DataIC50:  51nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50340001(CHEMBL1762478 | rac-4-chloro-2-(1-(methylamino)pen...)
Affinity DataIC50:  51nMAssay Description:Inhibition of human recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421056(CHEMBL2087846)
Affinity DataIC50:  54nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421067(CHEMBL2087858)
Affinity DataIC50:  55nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421057(CHEMBL2087847)
Affinity DataIC50:  56nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421068(CHEMBL2087859)
Affinity DataIC50:  57nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421044(CHEMBL2087622)
Affinity DataIC50:  60nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421069(CHEMBL2087860)
Affinity DataIC50:  62nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421058(CHEMBL2087848)
Affinity DataIC50:  63nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421059(CHEMBL2087849)
Affinity DataIC50:  69nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421070(CHEMBL2087861)
Affinity DataIC50:  70nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421071(CHEMBL2087862)
Affinity DataIC50:  70nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50339999((R)-2-(3-(methylamino)-1-phenylpropoxy)-4-(trifluo...)
Affinity DataIC50:  71nMAssay Description:Inhibition of human recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421060(CHEMBL2087850)
Affinity DataIC50:  72nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421072(CHEMBL2087863)
Affinity DataIC50:  74nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421088(CHEMBL2087851)
Affinity DataIC50:  79nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421073(CHEMBL2087864)
Affinity DataIC50:  80nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421045(CHEMBL2087623)
Affinity DataIC50:  86nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421043(CHEMBL2087621)
Affinity DataIC50:  87nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421074(CHEMBL2087865)
Affinity DataIC50:  88nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421080(CHEMBL2088115)
Affinity DataIC50:  89nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50124535(1-(6-CYANO-3-PYRIDYLCARBONYL)-5',8'-DIFLUOROSPIRO[...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50340000((R)-4-methoxy-2-(3-(methylamino)-1-phenylpropoxy)b...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421085(CHEMBL2088120)
Affinity DataIC50:  120nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421075(CHEMBL2087866)
Affinity DataIC50:  120nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421081(CHEMBL2088116)
Affinity DataIC50:  150nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421076(CHEMBL2087867)
Affinity DataIC50:  160nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421046(CHEMBL2087624)
Affinity DataIC50:  170nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421061(CHEMBL2087852)
Affinity DataIC50:  170nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421082(CHEMBL2088117)
Affinity DataIC50:  180nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Astrazeneca Charnwood

Curated by ChEMBL
LigandPNGBDBM50339998((R)-2-(3-amino-1-phenylpropylthio)-4-chlorobenzoni...)
Affinity DataIC50:  200nMAssay Description:Inhibition of iNOS in intact human DLD1 cells assessed as nitric oxide productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421062(CHEMBL2087853)
Affinity DataIC50:  220nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421047(CHEMBL2087625)
Affinity DataIC50:  220nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421048(CHEMBL2087626)
Affinity DataIC50:  220nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50421049(CHEMBL2087627)
Affinity DataIC50:  230nMAssay Description:Inhibition of Helicobacter pylori J99 glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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