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Found 14 with Last Name = 'keil' and Initial = 'r'
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50085072(1-{2-[(3-Fluoro-phenyl)-(4-fluoro-phenyl)-methoxy]...)
Affinity DataKi:  0.360nMAssay Description:Competitive binding versus [N-methyl-3H]-WIN 35,428 in murine kidney cells transfected with human dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50085071(3-(4-Iodo-phenyl)-6-methyl-6-aza-bicyclo[3.2.2]non...)
Affinity DataKi:  0.480nMAssay Description:In vitro affinity determined using [3H]-WIN- 35428 in murine kidney cells transfected with human dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50085071(3-(4-Iodo-phenyl)-6-methyl-6-aza-bicyclo[3.2.2]non...)
Affinity DataKi:  0.670nMAssay Description:In vitro affinity determined using [3H]-citalopram in murine kidney cells transfected with human serotonin transporter (SERT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50085069(3-(4-Chloro-phenyl)-6-methyl-6-aza-bicyclo[3.2.2]n...)
Affinity DataKi:  0.900nMAssay Description:Inhibition constant against [N-methyl-3H]-WIN 35428 in murine kidney cells transfected with human dopamine transporter.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM85616(MOLI000038 | [18F]FECNT)
Affinity DataKi:  1.53nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50028091((1E)-5-methoxy-1-[4-(trifluoromethyl)phenyl]pentan...)
Affinity DataKi:  3.08nMAssay Description:Inhibition constant against [3H]-citalopram in murine kidney cells transfected with human dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM85616(MOLI000038 | [18F]FECNT)
Affinity DataKi:  240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50085069(3-(4-Chloro-phenyl)-6-methyl-6-aza-bicyclo[3.2.2]n...)
Affinity DataKi:  427nMAssay Description:Inhibition constant against [3H]-citalopram in murine kidney cells transfected with human serotonin transporter.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Free University Of Berlin

Curated by ChEMBL
LigandPNGBDBM50409556(CHEMBL2068430)
Affinity DataEC50:  120nMAssay Description:Agonist activity in transcriptional activation assay in MCF-7-2a cells compared to estradiol E2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Free University Of Berlin

Curated by ChEMBL
LigandPNGBDBM50409553(CHEMBL112355)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity in transcriptional activation assay in MCF-7-2a cells compared to estradiol E2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Free University Of Berlin

Curated by ChEMBL
LigandPNGBDBM50409554(CHEMBL115729)
Affinity DataEC50:  620nMAssay Description:Agonist activity in transcriptional activation assay in MCF-7-2a cells compared to estradiol E2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Free University Of Berlin

Curated by ChEMBL
LigandPNGBDBM50116387(2-Chloro-4-[5-(2-chloro-4-hydroxy-phenyl)-4,5-dihy...)
Affinity DataEC50:  380nMAssay Description:Agonist activity in transcriptional activation assay in MCF-7-2a cells compared to estradiol E2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Free University Of Berlin

Curated by ChEMBL
LigandPNGBDBM50409555(CHEMBL323919)
Affinity DataEC50:  65nMAssay Description:Agonist activity in transcriptional activation assay in MCF-7-2a cells compared to estradiol E2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Free University Of Berlin

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  0.490nMAssay Description:Agonist activity in transcriptional activation assay in MCF-7-2a cells compared to estradiol E2More data for this Ligand-Target Pair