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Found 376 with Last Name = 'kiankarimi' and Initial = 'm'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190927(CHEMBL214513 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190919(CHEMBL386454 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50171332(1-(2-Bromo-4-isopropyl-phenyl)-7-methyl-5-(1-propy...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity for corticotropin-releasing factor-1 expressed in leukocyte tyrosine kinase cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190948(CHEMBL442064 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190943(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-N-((S)-1-(...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50171318(1-(4-Methoxy-phenyl)-7-methyl-5-(1-propyl-butyl)-4...)
Affinity DataKi:  2nMAssay Description:Binding affinity for corticotropin-releasing factor-1 expressed in leukocyte tyrosine kinase cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190931(CHEMBL265255 | N-((S)-1-((R)-3-(cyclopentylamino)p...)
Affinity DataKi:  2nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190922(5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-(tetrah...)
Affinity DataKi:  2nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190941(CHEMBL387013 | N-((S)-1-((R)-3-(3-cyclohexylpropyl...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190940(CHEMBL383933 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190929(5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-(methyl...)
Affinity DataKi:  3nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074501(Butyl-ethyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-ph...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity for corticotropin-releasing factor-1 expressed in leukocyte tyrosine kinase cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190918(CHEMBL215067 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190925(4'-Ethyl-biphenyl-4-carboxylic acid methyl-[(S)-1-...)
Affinity DataKi:  4nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190920(4'-ethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-...)
Affinity DataKi:  4nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190268(4'-methylsulfanyl-biphenyl-4-carboxylic acid methy...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50171325(2-(2,4-Dichloro-phenyl)-4-methyl-6-(1-propyl-butyl...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity for corticotropin-releasing factor-1 expressed in leukocyte tyrosine kinase cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190947(4'-ethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-...)
Affinity DataKi:  4.90nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190934(4'-ethyl-biphenyl-4-carboxylic acid methyl-{(S)-1-...)
Affinity DataKi:  5nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190921(CHEMBL267797 | N-((S)-1-((R)-3-(dimethylamino)pyrr...)
Affinity DataKi:  5nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50171322(1-(2,4-Dichloro-phenyl)-7-methyl-5-(1-propyl-butyl...)
Affinity DataKi:  5.10nMAssay Description:Binding affinity for corticotropin-releasing factor-1 expressed in leukocyte tyrosine kinase cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190932(4'-methoxy-2'-methyl-biphenyl-4-carboxylic acid {(...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190279(4'-chloro-biphenyl-4-carboxylic acid methyl-{(S)-1...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190944(5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-(methyl...)
Affinity DataKi:  6nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190280(4'-trifluoromethoxy-biphenyl-4-carboxylic acid met...)
Affinity DataKi:  7nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190933(5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-((tetra...)
Affinity DataKi:  8nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50171316(5-(1-Ethyl-propyl)-1-(4-methoxy-phenyl)-7-methyl-4...)
Affinity DataKi:  8nMAssay Description:Binding affinity for corticotropin-releasing factor-1 expressed in leukocyte tyrosine kinase cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190267(4'-methoxy-biphenyl-4-carboxylic acid methyl-{(S)-...)
Affinity DataKi:  8nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190296(4'-trifluoromethyl-biphenyl-4-carboxylic acid meth...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190936(5-(4-methoxyphenyl)-N-methyl-N-((S)-1-((R)-3-(tetr...)
Affinity DataKi:  10nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190939(4'-ethyl-biphenyl-4-carboxylic acid [(S)-1-((R)-3-...)
Affinity DataKi:  11nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190938(5-(4-ethylphenyl)-N-((S)-1-((R)-3-(isopropylamino)...)
Affinity DataKi:  11nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190293(4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190263(4'-trifluoromethyl-biphenyl-4-carboxylic acid meth...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190281(4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50171328(1-(4-Chloro-phenyl)-7-methyl-5-(1-propyl-butyl)-4,...)
Affinity DataKi:  12nMAssay Description:Binding affinity for corticotropin-releasing factor-1 expressed in leukocyte tyrosine kinase cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190261(4'-trifluoromethyl-biphenyl-4-carboxylic acid meth...)
Affinity DataKi:  13nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190290(4'-trifluoromethyl-biphenyl-4-carboxylic acid ((S)...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190935(4'-ethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-...)
Affinity DataKi:  14nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190303(4'-trifluoromethyl-biphenyl-4-carboxylic acid [(S)...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190274(4'-trifluoromethyl-biphenyl-4-carboxylic acid meth...)
Affinity DataKi:  16nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190923(CHEMBL386969 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  16nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190291(4'-trifluoromethyl-biphenyl-4-carboxylic acid meth...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50171334(7-Methyl-5-(1-propyl-butyl)-1-(4-trifluoromethyl-p...)
Affinity DataKi:  17nMAssay Description:Binding affinity for corticotropin-releasing factor-1 expressed in leukocyte tyrosine kinase cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190930(4'-ethyl-biphenyl-4-carboxylic acid [(S)-1-((R)-3-...)
Affinity DataKi:  18nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190297(4'-trifluoromethyl-biphenyl-4-carboxylic acid ((S)...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190272(4'-fluoro-biphenyl-4-carboxylic acid methyl-{(S)-1...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50171321(5-(1-Ethyl-propyl)-1-(4-methoxy-2-methyl-phenyl)-7...)
Affinity DataKi:  20nMAssay Description:Binding affinity for corticotropin-releasing factor-1 expressed in leukocyte tyrosine kinase cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190928(CHEMBL384234 | N-((S)-1-((R)-3-(3-cyclohexylpropyl...)
Affinity DataKi:  21nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190302(4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)...)
Affinity DataKi:  21nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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