Affinity DataKi: 5.10nMAssay Description:TP_TRANSPORTER: inhibition of Dopamine uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:TP_TRANSPORTER: inhibition of Adrenaline uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:TP_TRANSPORTER: inhibition of Noradrenaline uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:TP_TRANSPORTER: inhibition of Serotonin uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:TP_TRANSPORTER: inhibition of Dopamine uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:TP_TRANSPORTER: inhibition of Adrenaline uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:TP_TRANSPORTER: inhibition of Noradrenaline uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 605nMAssay Description:TP_TRANSPORTER: inhibition of Serotonin uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg
Curated by ChEMBL
University Of Heidelberg
Curated by ChEMBL
Affinity DataKi: 1.40E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.90E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+6nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair