Affinity DataKi: 1nM ΔG°: -53.4kJ/mole IC50: 5nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity of the compound against HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Binding affinity of the compound against HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:Binding affinity of the compound against HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Binding affinity of the compound against HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nM ΔG°: >-23.7kJ/mole IC50: >1.00E+5nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Gilead Sciences
Curated by ChEMBL
Gilead Sciences
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Concentration needed to inhibit HIV- protease activity by 50%.More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMAssay Description:Inhibitory activity against Methionine aminopeptidase 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Inhibitory activity against Methionine aminopeptidase 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 0.510nMAssay Description:Inhibitory activity against Methionine aminopeptidase 2More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Gilead Sciences
Curated by ChEMBL
Gilead Sciences
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Concentration needed to inhibit HIV- protease activity by 50%.More data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Inhibitory activity against Methionine aminopeptidase 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibitory activity against Methionine aminopeptidase 2More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Gilead Sciences
Curated by ChEMBL
Gilead Sciences
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Concentration needed to inhibit HIV- protease activity by 50%.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against Methionine aminopeptidase 2More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against Methionine aminopeptidase 2More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibitory activity against Methionine aminopeptidase 2More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of neuraminidase of influenza A/PR/8/34(H1N1)More data for this Ligand-Target Pair
TargetGenome polyprotein [1027-1657](Hepatitis C virus genotype 1a (isolate 1) (HCV))
Gilead Sciences
US Patent
Gilead Sciences
US Patent
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using HCV protease.More data for this Ligand-Target Pair
TargetGenome polyprotein [1027-1657](Hepatitis C virus genotype 1a (isolate 1) (HCV))
Gilead Sciences
US Patent
Gilead Sciences
US Patent
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using HCV protease.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
TargetGenome polyprotein [1027-1657](Hepatitis C virus genotype 1a (isolate 1) (HCV))
Gilead Sciences
US Patent
Gilead Sciences
US Patent
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using HCV protease.More data for this Ligand-Target Pair
TargetGenome polyprotein [1027-1657](Hepatitis C virus genotype 1a (isolate 1) (HCV))
Gilead Sciences
US Patent
Gilead Sciences
US Patent
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using HCV protease.More data for this Ligand-Target Pair
TargetGenome polyprotein [1027-1657](Hepatitis C virus genotype 1a (isolate 1) (HCV))
Gilead Sciences
US Patent
Gilead Sciences
US Patent
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using HCV protease.More data for this Ligand-Target Pair
TargetGenome polyprotein [1027-1657](Hepatitis C virus genotype 1a (isolate 1) (HCV))
Gilead Sciences
US Patent
Gilead Sciences
US Patent
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using HCV protease.More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
TargetGenome polyprotein [1027-1657](Hepatitis C virus genotype 1a (isolate 1) (HCV))
Gilead Sciences
US Patent
Gilead Sciences
US Patent
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using HCV protease.More data for this Ligand-Target Pair
TargetGenome polyprotein [1027-1657](Hepatitis C virus genotype 1a (isolate 1) (HCV))
Gilead Sciences
US Patent
Gilead Sciences
US Patent
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using HCV protease.More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
TargetGenome polyprotein [1027-1657](Hepatitis C virus genotype 1a (isolate 1) (HCV))
Gilead Sciences
US Patent
Gilead Sciences
US Patent
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using HCV protease.More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair