TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
University Of Science And Technology
Curated by ChEMBL
University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human His6-tagged full length PRL3 assessed as inhibition of DiFMUP dephosphorylationMore data for this Ligand-Target Pair
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
University Of Science And Technology
Curated by ChEMBL
University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human His6-tagged full length PRL3 assessed as inhibition of DiFMUP dephosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 1.64E+4nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 3.22E+4nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 5.27E+4nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 7.10E+4nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair