Compile Data Set for Download or QSAR
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Found 149 with Last Name = 'kiyoi' and Initial = 'y'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418229(CHEMBL1760646)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418228(CHEMBL1760645)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  0.933nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418210(CHEMBL1760664)
Affinity DataKi:  4.37nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418212(CHEMBL1760663)
Affinity DataKi:  5.01nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418213(CHEMBL1760661)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418211(CHEMBL1760662)
Affinity DataKi:  7.59nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  851nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418210(CHEMBL1760664)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418229(CHEMBL1760646)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418228(CHEMBL1760645)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418222(CHEMBL1760652)
Affinity DataIC50:  0.513nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418221(CHEMBL1760653)
Affinity DataIC50:  0.575nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418220(CHEMBL1760654)
Affinity DataIC50:  0.631nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418223(CHEMBL1760651)
Affinity DataIC50:  0.759nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418224(CHEMBL1760650)
Affinity DataIC50:  0.776nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543723(CHEMBL4640512)
Affinity DataIC50:  1nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418229(CHEMBL1760646)
Affinity DataIC50:  1.17nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418217(CHEMBL1760657)
Affinity DataIC50:  1.32nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418216(CHEMBL1760658)
Affinity DataIC50:  1.48nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418206(CHEMBL1760668)
Affinity DataIC50:  1.48nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418219(CHEMBL1760655)
Affinity DataIC50:  1.55nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418228(CHEMBL1760645)
Affinity DataIC50:  1.82nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418225(CHEMBL1760649)
Affinity DataIC50:  2nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543691(CHEMBL4646369)
Affinity DataIC50:  2nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418215(CHEMBL1760659)
Affinity DataIC50:  2.57nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418205(CHEMBL1760669)
Affinity DataIC50:  2.63nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543711(CHEMBL4632660)
Affinity DataIC50:  3nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543712(CHEMBL4642115)
Affinity DataIC50:  4nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418214(CHEMBL1760660)
Affinity DataIC50:  4.90nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543692(CHEMBL4635996)
Affinity DataIC50:  5nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418210(CHEMBL1760664)
Affinity DataIC50:  5.13nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418218(CHEMBL1760656)
Affinity DataIC50:  5.13nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418203(CHEMBL1760644)
Affinity DataIC50:  5.13nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418226(CHEMBL1760648)
Affinity DataIC50:  5.37nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543689(CHEMBL4637782)
Affinity DataIC50:  6nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543690(CHEMBL4636658)
Affinity DataIC50:  6nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418207(CHEMBL1760667)
Affinity DataIC50:  6.03nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543695(CHEMBL4649886)
Affinity DataIC50:  7nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418208(CHEMBL1760666)
Affinity DataIC50:  8.13nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418227(CHEMBL1760647)
Affinity DataIC50:  8.32nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418209(CHEMBL1760665)
Affinity DataIC50:  8.91nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543696(CHEMBL4649330)
Affinity DataIC50:  9nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418204(CHEMBL1760670)
Affinity DataIC50:  9.33nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543717(CHEMBL4639651)
Affinity DataIC50:  10nMAssay Description:Inhibition of factor 11a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50:  11.2nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418211(CHEMBL1760662)
Affinity DataIC50:  11.5nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543719(CHEMBL4646710)
Affinity DataIC50:  12nMAssay Description:Inhibition of factor 11a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418212(CHEMBL1760663)
Affinity DataIC50:  13.5nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50543720(CHEMBL4646911)
Affinity DataIC50:  15nMAssay Description:Inhibition of factor 11a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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