Compile Data Set for Download or QSAR
maximum 50k data
Found 60 with Last Name = 'kolusheva' and Initial = 's'
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50244449((E)-(2-(hydroxymethyl)-4-((1-methyl-1H-indol-3-yl)...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50244449((E)-(2-(hydroxymethyl)-4-((1-methyl-1H-indol-3-yl)...)
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017890(CHEMBL3289012)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017890(CHEMBL3289012)
Affinity DataKi:  0.410nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017892(CHEMBL3289014)
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017891(CHEMBL3289013)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017892(CHEMBL3289014)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017891(CHEMBL3289013)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017889(CHEMBL3289011)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017889(CHEMBL3289011)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017890(CHEMBL3289012)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50017891(CHEMBL3289013)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017891(CHEMBL3289013)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50017890(CHEMBL3289012)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017892(CHEMBL3289014)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50017892(CHEMBL3289014)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017889(CHEMBL3289011)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50244449((E)-(2-(hydroxymethyl)-4-((1-methyl-1H-indol-3-yl)...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50017889(CHEMBL3289011)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50244449((E)-(2-(hydroxymethyl)-4-((1-methyl-1H-indol-3-yl)...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 60 total ) | Next | Last >>
Jump to: