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Found 168 with Last Name = 'komatsu' and Initial = 'k'
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395262(CHEMBL2163999)
Affinity DataKi:  6.00E+3nMAssay Description:Competitive inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395284(CHEMBL2163996)
Affinity DataIC50:  3nMAssay Description:Inhibition of CDK2 after 60 mins using [33P]-gamma-ATP by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395283(CHEMBL2163995)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of CDK2 after 60 mins using [33P]-gamma-ATP by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395285(CHEMBL2163997)
Affinity DataIC50:  4nMAssay Description:Inhibition of CDK2 after 60 mins using [33P]-gamma-ATP by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209796(CHEMBL3885011)
Affinity DataIC50:  5nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395272(CHEMBL1231206)
Affinity DataIC50:  5nMAssay Description:Binding affinity to recombinant MAPKAP-K2 using KKKALSRQLSVAA as substrate after 4 mins by surface plasmon resonance spectroscopic analysisMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209789(CHEMBL3885174)
Affinity DataIC50:  10nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209788(CHEMBL3884506)
Affinity DataIC50:  22nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209791(CHEMBL3883560)
Affinity DataIC50:  32nMAssay Description:Inhibition of HDAC2 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209791(CHEMBL3883560)
Affinity DataIC50:  33nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209789(CHEMBL3885174)
Affinity DataIC50:  35nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209794(CHEMBL3884118)
Affinity DataIC50:  49nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209790(CHEMBL3885367)
Affinity DataIC50:  49nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209834(CHEMBL3884141)
Affinity DataIC50:  50nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209797(CHEMBL3885245)
Affinity DataIC50:  50nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395267(CHEMBL2163608)
Affinity DataIC50:  54nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395262(CHEMBL2163999)
Affinity DataIC50:  55nMAssay Description:Inhibition of CDK2 after 60 mins using [33P]-gamma-ATP by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395269(CHEMBL2163610)
Affinity DataIC50:  57nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209788(CHEMBL3884506)
Affinity DataIC50:  59nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209791(CHEMBL3883560)
Affinity DataIC50:  60nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209829(CHEMBL3883830)
Affinity DataIC50:  61nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209835(CHEMBL3885496)
Affinity DataIC50:  66nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395268(CHEMBL2163611)
Affinity DataIC50:  76nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209795(CHEMBL3884044)
Affinity DataIC50:  76nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209792(CHEMBL3884279)
Affinity DataIC50:  83nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209789(CHEMBL3885174)
Affinity DataIC50:  89nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209787(CHEMBL3883667)
Affinity DataIC50:  92nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209790(CHEMBL3885367)
Affinity DataIC50:  109nMAssay Description:Inhibition of HDAC8 (unknown origin) after 2.5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209788(CHEMBL3884506)
Affinity DataIC50:  111nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209788(CHEMBL3884506)
Affinity DataIC50:  116nMAssay Description:Inhibition of HDAC8 (unknown origin) after 2.5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395274(CHEMBL1235213)
Affinity DataIC50:  130nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395275(CHEMBL2163616)
Affinity DataIC50:  130nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50225787(2,4-diamino-6,7-dihydroxy-10H-9-oxa-1-aza-anthrace...)
Affinity DataIC50:  130nMAssay Description:Inhibition of MAPKAP-K2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209789(CHEMBL3885174)
Affinity DataIC50:  135nMAssay Description:Inhibition of HDAC8 (unknown origin) after 2.5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395270(CHEMBL2163609)
Affinity DataIC50:  140nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395271(CHEMBL2163612)
Affinity DataIC50:  160nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209834(CHEMBL3884141)
Affinity DataIC50:  163nMAssay Description:Inhibition of HDAC2 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209796(CHEMBL3885011)
Affinity DataIC50:  181nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209791(CHEMBL3883560)
Affinity DataIC50:  183nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209787(CHEMBL3883667)
Affinity DataIC50:  191nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma

Curated by ChEMBL
LigandPNGBDBM50395266(CHEMBL2163607)
Affinity DataIC50:  200nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209792(CHEMBL3884279)
Affinity DataIC50:  208nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209796(CHEMBL3885011)
Affinity DataIC50:  209nMAssay Description:Inhibition of HDAC2 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209798(CHEMBL3884552)
Affinity DataIC50:  224nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209795(CHEMBL3884044)
Affinity DataIC50:  226nMAssay Description:Inhibition of HDAC8 (unknown origin) after 2.5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209787(CHEMBL3883667)
Affinity DataIC50:  232nMAssay Description:Inhibition of HDAC2 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209796(CHEMBL3885011)
Affinity DataIC50:  251nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209829(CHEMBL3883830)
Affinity DataIC50:  256nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209834(CHEMBL3884141)
Affinity DataIC50:  261nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50209797(CHEMBL3885245)
Affinity DataIC50:  283nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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