Affinity DataKi: 6.00E+3nMAssay Description:Competitive inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK2 after 60 mins using [33P]-gamma-ATP by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of CDK2 after 60 mins using [33P]-gamma-ATP by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2 after 60 mins using [33P]-gamma-ATP by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to recombinant MAPKAP-K2 using KKKALSRQLSVAA as substrate after 4 mins by surface plasmon resonance spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of HDAC2 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of CDK2 after 60 mins using [33P]-gamma-ATP by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 109nMAssay Description:Inhibition of HDAC8 (unknown origin) after 2.5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 111nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 116nMAssay Description:Inhibition of HDAC8 (unknown origin) after 2.5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of MAPKAP-K2More data for this Ligand-Target Pair
Affinity DataIC50: 135nMAssay Description:Inhibition of HDAC8 (unknown origin) after 2.5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 163nMAssay Description:Inhibition of HDAC2 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 181nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 183nMAssay Description:Inhibition of HDAC6 (unknown origin) after 20 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 191nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 208nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 209nMAssay Description:Inhibition of HDAC2 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 224nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 226nMAssay Description:Inhibition of HDAC8 (unknown origin) after 2.5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 232nMAssay Description:Inhibition of HDAC2 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 256nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 261nMAssay Description:Inhibition of HDAC1 (unknown origin) after 24 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 283nMAssay Description:Inhibition of HDAC3 (unknown origin) after 5 hrs by SAMDI mass spectroscopic analysisMore data for this Ligand-Target Pair