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Found 116 with Last Name = 'kopcho' and Initial = 'j'
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090867((2R,3S,4R,5R)-2-(aminomethyl)-5-(4-chloro-5-iodo-7...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090843((1R,5S)-2-((3R,4aR)-4-Amino-5-bromo-pyrrolo[2,3-d]...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174602((4R,5R,6S)-5-[4-(4-Fluoro-phenylamino)-5-phenyl-py...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134740((1R,4S,5R)-2-Hydroxymethyl-5-(5-phenyl-4-phenylami...)
Affinity DataIC50:  0.470nMAssay Description:Inhibitory activity against human recombinant adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134740((1R,4S,5R)-2-Hydroxymethyl-5-(5-phenyl-4-phenylami...)
Affinity DataIC50:  0.470nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090887((1R,4S,5R)-2-Methyl-5-(5-phenyl-4-phenylamino-pyrr...)
Affinity DataIC50:  0.5nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090887((1R,4S,5R)-2-Methyl-5-(5-phenyl-4-phenylamino-pyrr...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090862((1R,5S)-2-((3R,4aR)-4-Amino-5-iodo-pyrrolo[2,3-d]p...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134753((1R,4S,5R)-2-Methyl-5-(5-phenyl-4-phenylamino-pyrr...)
Affinity DataIC50:  0.800nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134753((1R,4S,5R)-2-Methyl-5-(5-phenyl-4-phenylamino-pyrr...)
Affinity DataIC50:  0.800nMAssay Description:Inhibitory activity against human recombinant adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090883((1R,4S,5R)-2-Hydroxymethyl-5-(5-phenyl-4-phenylami...)
Affinity DataIC50:  0.800nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090883((1R,4S,5R)-2-Hydroxymethyl-5-(5-phenyl-4-phenylami...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090874(2-[4-(4-Hydroxy-phenylamino)-5-phenyl-pyrrolo[2,3-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090880(4-[7-(3,4-Dihydroxy-5-methyl-tetrahydro-furan-2-yl...)
Affinity DataIC50:  1nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090881((2R,3R,4S,5R)-2-(6-Bromo-5-phenyl-4-phenylamino-py...)
Affinity DataIC50:  1nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174603((1R,2R,3R)-2-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl...)
Affinity DataIC50:  1nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090875(2-[5-(4-Chloro-phenyl)-4-phenylamino-pyrrolo[2,3-d...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090900(2-Azidomethyl-5-(5-phenyl-4-phenylamino-pyrrolo[2,...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090901(2-Methyl-5-(5-phenyl-4-p-tolylamino-pyrrolo[2,3-d]...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090895((2R,3R,4S,5R)-2-[4-(4-Fluoro-phenylamino)-5-phenyl...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134756((2S,3S,4R,5R)-2-[4-(4-Fluoro-phenylamino)-5-phenyl...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory activity against human recombinant adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174591(4-[7-((1R,2R,3R)-3,4-Dihydroxy-tetrahydro-furan-2-...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174594((1R,2R,3R)-2-[4-(3-Ethoxy-phenylamino)-5-phenyl-py...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090889(2-[4-(4-Chloro-phenylamino)-5-phenyl-pyrrolo[2,3-d...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090899(2-[5-(4-Chloro-phenyl)-4-(4-chloro-phenylamino)-py...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134751((2R,3R,4S,5S)-2-Hydroxymethyl-5-(3-phenyl-4-phenyl...)
Affinity DataIC50:  2.80nMAssay Description:Inhibitory activity against human recombinant adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174599((1R,2R,3R)-2-[4-(4-Ethoxy-phenylamino)-5-phenyl-py...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090844((2R,3R,4S,5R)-2-(4-Chloro-5-iodo-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  3nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090884(2-(5-Furan-2-yl-4-phenylamino-pyrrolo[2,3-d]pyrimi...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134744((2S,3S,4R,5S)-2-(4-Amino-3-bromo-pyrazolo[3,4-d]py...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against human recombinant adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174593((1R,2R,3R)-2-(5-Phenyl-4-phenylamino-pyrrolo[2,3-d...)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174598((1R,2R,3R)-2-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl...)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174597((1R,2R,3R)-2-[4-(4-Bromo-phenylamino)-5-phenyl-pyr...)
Affinity DataIC50:  5nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090895((2R,3R,4S,5R)-2-[4-(4-Fluoro-phenylamino)-5-phenyl...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against human recombinant adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174600((1R,2R,3R)-2-[5-(4-Ethoxy-phenyl)-4-(2-methoxy-phe...)
Affinity DataIC50:  5.30nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174592((1R,2R,3R)-2-(4-Amino-5-iodo-pyrrolo[2,3-d]pyrimid...)
Affinity DataIC50:  6nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174596((1R,2R,3R)-2-[4-(4-Fluoro-phenylamino)-5-phenyl-py...)
Affinity DataIC50:  6nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090893(2-[4-(4-Methoxy-phenylamino)-5-phenyl-pyrrolo[2,3-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090897(2-Aminomethyl-5-(5-phenyl-4-phenylamino-pyrrolo[2,...)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174605(4-[5-(4-Chloro-phenyl)-7-((1R,2R,3R)-3,4-dihydroxy...)
Affinity DataIC50:  7nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090898(2-[5-Furan-2-yl-4-(4-methoxy-phenylamino)-pyrrolo[...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090854((2R,3S,4R,5R)-2-(azidomethyl)-5-(4-chloro-5-iodo-7...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM14486((2R,3R,4S,5R)-2-(2-amino-9-iodo-3,5,7-triazabicycl...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM14486((2R,3R,4S,5R)-2-(2-amino-9-iodo-3,5,7-triazabicycl...)
Affinity DataIC50:  9nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50174601((1R,2R,3R)-2-[5-(3-Amino-phenyl)-4-(4-fluoro-pheny...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090890(4-[7-(3,4-Dihydroxy-5-methyl-tetrahydro-furan-2-yl...)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134745((2R,3R,4S,5S)-2-Methoxymethyl-5-(5-phenyl-4-phenyl...)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity against human recombinant adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134743((2S,3S,4R,5R)-2-(4-Amino-5-iodo-pyrrolo[2,3-d]pyri...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity against human recombinant adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090853((2R,3R,4S,5R)-2-(4-Chloro-5-iodo-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  24nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50090891(2-Methyl-5-[5-phenyl-4-(pyridin-3-ylamino)-pyrrolo...)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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