Affinity DataKi: 27nMAssay Description:Inhibition of Flaveria bidentis carbonic anhydrase 1 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Inhibition of Saccharomyces cerevisiae carbonic anhydrase SceCA preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.76E+3nMAssay Description:Mixed-type inhibition of equine serum BChE using S-butyrylthiocholine chloride as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.21E+4nMAssay Description:Inhibition of Methanobacterium thermoautotrophicum beta-carbonic anhydrase preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 920nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of horse serum BChE using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of human Protein kinase C gammaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibition of Protein kinase C beta 2More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide substrate by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of Protein kinase C epsilonMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.24E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of horse serum BChE using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.68E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
Affinity DataIC50: 2.86E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
Affinity DataIC50: 2.91E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair