Affinity DataKi: 0.790nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serotonin (5-HT) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 1.06nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serototnin (5-HT) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 3.66nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serototnin (5-HT) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 4.72nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 7.45nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serototnin (5-HT) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 18.4nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 63.9nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serototnin (5-HT) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 97.1nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serotonin (5-HT) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 163nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 235nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Ability to inhibit [3H]-WIN-35,428 binding to cloned human dopamine (DA) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 266nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serotonin (5-HT) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 353nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporter; Average of two experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 695nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 695nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serotonin (5-HT) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 920nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 1.45E+3nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serotonin (5-HT) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 2.81E+3nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 3.11E+3nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serotonin (5-HT) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+3nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 5.45E+3nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporterMore data for this Ligand-Target Pair
Affinity DataKi: 7.27E+3nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serotonin (5-HT) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serotonin (5-HT) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-paroxetine binding to cloned human serotonin (5-HT) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-nisoxatine binding to cloned human norepinephrine (NE) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporterMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to inhibit [3H]-mazindol binding to cloned human dopamine (DA) transporterMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.0430nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.0430nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.0780nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.0780nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.133nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.133nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.145nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.145nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.214nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.214nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.218nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair