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Found 28 with Last Name = 'kutz' and Initial = 'cj'
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50464671(CHEMBL3621615)
Affinity DataKi:  2.20E+3nMAssay Description:Competitive inhibition of LSD1 (unknown origin) incubated for 30 mins using H3K4me2 substrate by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50065386(CHEMBL3401327)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of human recombinant LSD1 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetREST corepressor 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50464671(CHEMBL3621615)
Affinity DataIC50:  1.19E+3nMAssay Description:Inhibition of recombinant LSD1/CoREST (unknown origin) assessed as residual activity for 30 mins to 4 hrs by fluorescence based assay relative to con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetREST corepressor 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50498660(CHEMBL1605826)
Affinity DataIC50:  2.22E+3nMAssay Description:Inhibition of recombinant LSD1/CoREST (unknown origin) assessed as residual activity for 30 mins to 4 hrs by fluorescence based assay relative to con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
John Hopkins University

Curated by ChEMBL
LigandPNGBDBM50113851((+/-)-Tranylcypromine | 2-PCPA | 2-Phenyl-cyclopro...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of MAO-A (unknown origin) by MAo-Glo kit analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
John Hopkins University

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | CHEMBL25799...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of MAOA (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50065386(CHEMBL3401327)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of human recombinant LSD1 after 30 mins to 4 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | CHEMBL25799...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of MAOB (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50113851((+/-)-Tranylcypromine | 2-PCPA | 2-Phenyl-cyclopro...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of MAO-B (unknown origin) by MAo-Glo kit analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50065385(CHEMBL3401326)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human recombinant LSD1 after 30 mins to 4 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50065384(CHEMBL3401325)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human recombinant LSD1 after 30 mins to 4 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50065382(CHEMBL1085949)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of MAO-B (unknown origin) by MAo-Glo kit analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50065382(CHEMBL1085949)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human recombinant LSD1 after 30 mins to 4 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50065383(CHEMBL3144164)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human recombinant LSD1 after 30 mins to 4 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50065386(CHEMBL3401327)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of MAO-B (unknown origin) by MAo-Glo kit analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetREST corepressor 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | CHEMBL25799...)
Affinity DataIC50:  2.07E+4nMAssay Description:Inhibition of recombinant LSD1/CoREST (unknown origin) assessed as residual activity for 30 mins to 4 hrs by fluorescence based assay relative to con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50065385(CHEMBL3401326)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of MAO-B (unknown origin) by MAo-Glo kit analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50065384(CHEMBL3401325)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of MAO-B (unknown origin) by MAo-Glo kit analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
John Hopkins University

Curated by ChEMBL
LigandPNGBDBM50065382(CHEMBL1085949)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of MAO-A (unknown origin) by MAo-Glo kit analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
John Hopkins University

Curated by ChEMBL
LigandPNGBDBM50065384(CHEMBL3401325)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-A (unknown origin) by MAo-Glo kit analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
John Hopkins University

Curated by ChEMBL
LigandPNGBDBM50065386(CHEMBL3401327)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-A (unknown origin) by MAo-Glo kit analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50498660(CHEMBL1605826)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAOB (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
John Hopkins University

Curated by ChEMBL
LigandPNGBDBM50464671(CHEMBL3621615)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAOA (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
John Hopkins University

Curated by ChEMBL
LigandPNGBDBM50065385(CHEMBL3401326)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-A (unknown origin) by MAo-Glo kit analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
John Hopkins University

Curated by ChEMBL
LigandPNGBDBM50498660(CHEMBL1605826)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAOA (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50464671(CHEMBL3621615)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAOB (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50113851((+/-)-Tranylcypromine | 2-PCPA | 2-Phenyl-cyclopro...)
Affinity DataIC50:  2.42E+5nMAssay Description:Inhibition of human recombinant LSD1 after 30 mins to 4 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50113851((+/-)-Tranylcypromine | 2-PCPA | 2-Phenyl-cyclopro...)
Affinity DataIC50:  2.42E+5nMAssay Description:Irreversible inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed