Compile Data Set for Download or QSAR
maximum 50k data
Found 411 with Last Name = 'lamotte' and Initial = 'y'
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50043280(4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidaz...)
Affinity DataIC50:  3nMAssay Description:Inhibition of AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50306508(4'-((2,3-dimethyl-5-(1-phenylpropylcarbamoyl)-1H-i...)
Affinity DataIC50:  8nMAssay Description:Displacement of radiolabled ((5-{4-[Methyl-pyridin-2yl-amino)-ethoxy]-benzyl}-thiazolidine-2,4-dione) from human PPARgamma ligand binding domain expr...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634316(8,14-dioxa-4,10,19,20- | US20230357269, Example 1)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634318(4-fluoro-8,14-dioxa-10,19,20- | US20230357269, Exa...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634319(8,14-dioxa-10,19,20,23- | US20230357269, Example 4)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634320(8,14-dioxa-10,19,20- | US20230357269, Example 5)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634322(8,14-dioxa-5,10,19,20- | US20230357269, Example 7)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634323(4-methoxy-8,14-dioxa-10,19,20- | US20230357269, Ex...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634324(4-bromo-8,14-dioxa-10,19,20- | US20230357269, Exam...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634325(5-fluoro-8,14-dioxa-10,19,20- | US20230357269, Exa...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634326(5-methyl-8,14-dioxa-10,19,20- | US20230357269, Exa...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634327(4-(pyrrolidin-1-yl)-8,14-dioxa-10,19,20- | US20230...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634328(4-[4-(propan-2-yl)piperazin-1-yl]-8,14-dioxa- | US...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM50580006(CHEMBL5090730 | US20230357269, Example 14)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM50580007(CHEMBL5072941 | US20230357269, Example 15)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634331(4-(morpholin-4-yl)-8,14-dioxa-10,19,20- | US202303...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634332(4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-8,14- | US2...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634333(4-methyl-8,14-dioxa-10,19,20- | US20230357269, Exa...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634334(5-methoxy-8,14-dioxa-10,19,20- | US20230357269, Ex...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634335(4-(4,4-difluoropiperidin-1-yl)-8,14-dioxa- | US202...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634336(4-(3,3-difluoropyrrolidin-1-yl)-8,14-dioxa- | US20...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634337(7-methyl-8,14-dioxa-10,19,20- | US20230357269, Exa...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634338(4-[4-(2-methoxyethyl)piperidin-1-yl]-8,14-dioxa- |...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634340(4-[(3R)-3-hydroxypyrrolidin-1-yl]-8,14-dioxa- | US...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634341(4-[(2-methoxyethyl)(methyl)amino]-8,14-dioxa- | US...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634342(4-chloro-8,14-dioxa-10,19,20- | US20230357269, Exa...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634343(4-fluoro-5-methyl-8,14-dioxa-10,19,20- | US2023035...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634344(4,5-difluoro-8,14-dioxa-10,19,20- | US20230357269,...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634345(5-bromo-8,14-dioxa-10,19,20- | US20230357269, Exam...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634346(4-(4-methylpiperazin-1-yl)-8,14-dioxa-10,19,20- | ...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634347(4-(3-methoxyazetidin-1-yl)-8,14-dioxa-10,19,20- | ...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634348(1-{9-oxo-8,14-dioxa-10,19,20-triazatetra | US20230...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM50580008(CHEMBL5093627 | US20230357269, Example 34)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634350(4-(azetidin-1-yl)-8,14-dioxa-10,19,20- | US2023035...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634351(4-(piperidin-1-yl)-8,14-dioxa-10,19,20- | US202303...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634352(4-(2,5-dihydrofuran-3-yl)-8,14-dioxa-10,19,20- | U...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM50580009(CHEMBL5082872 | US20230357269, Example 38)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634354(4-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)-8,14- ...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634355(4-[(2S,5S)-2,5-dimethylmorpholin-4-yl]-8,14- | US2...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634356(4-[(morpholin-4-yl)methyl]-8,14-dioxa-10,19,20- | ...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634357(4-[(pyrrolidin-1-yl)methyl]-8,14-dioxa-10,19,20- |...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634359(4-[(4-methylpiperazin-1-yl)methyl]-8,14-dioxa- | U...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634360(5-(morpholin-4-yl)-8,14-dioxa-10,19,20- | US202303...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634361(4-[4-(2-methoxyethyl)piperazin-1-yl]-8,14-dioxa- |...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634362(4-(diethylamino)-8,14-dioxa-10,19,20-triazatetracy...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634363(4-cyclopropyl-8,14-dioxa-10,19,20- | US20230357269...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634365(13-methyl-8,14-dioxa-10,19,20- | US20230357269, Ex...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634366(8,14-dioxa-4,5,10,19,20- | US20230357269, Example ...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634367(4-[methyl(oxetan-3-yl)amino]-8,14-dioxa- | US20230...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Les Laboratoires Servier

US Patent
LigandPNGBDBM634369(4,10-dimethyl-8,14-dioxa-10,19,20- | US20230357269...)
Affinity DataIC50: <10nMAssay Description:LRRK2 Kinase reactions were carried out in 384-well white polystyrene plates in a final volume of 6 μl using ADP-Glo Kinase Assay kit (Promega C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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