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Found 30 with Last Name = 'le baut' and Initial = 'g'
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50179635((+)-5-[(4-chlorophenyl)(1H-imidazol-1-yl)methyl]-1...)
Affinity DataIC50:  9nMAssay Description:Inhibition of CYP19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50179635((+)-5-[(4-chlorophenyl)(1H-imidazol-1-yl)methyl]-1...)
Affinity DataIC50:  9nMAssay Description:Inhibition of CYP19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50179635((+)-5-[(4-chlorophenyl)(1H-imidazol-1-yl)methyl]-1...)
Affinity DataIC50:  15.3nMAssay Description:Inhibition of CYP19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50179639(4-((1H-imidazol-1-yl)(1H-indol-5-yl)methyl)benzoni...)
Affinity DataIC50:  19.3nMAssay Description:Inhibition of CYP19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50179637(5-((4-chlorophenyl)(1H-imidazol-1-yl)methyl)-1-met...)
Affinity DataIC50:  23.7nMAssay Description:Inhibition of CYP19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50179636(5-((4-fluorophenyl)(1H-imidazol-1-yl)methyl)-1H-in...)
Affinity DataIC50:  26.3nMAssay Description:Inhibition of CYP19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50179638(5-((3-chlorophenyl)(1H-imidazol-1-yl)methyl)-1H-in...)
Affinity DataIC50:  29.7nMAssay Description:Inhibition of CYP19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50075009(1-Ethyl-5-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50:  40nMAssay Description:Inhibition of CYP19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50075009(1-Ethyl-5-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50:  41nMAssay Description:In vitro inhibition of human Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50075009(1-Ethyl-5-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50:  41nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50075001(4-(3-Imidazol-1-ylmethyl-indol-1-ylmethyl)-benzoni...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibition of human Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50075003(5-Bromo-1-ethyl-3-[(4-fluoro-phenyl)-imidazol-1-yl...)
Affinity DataIC50:  52nMAssay Description:In vitro inhibition of human Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50075008(1-(2-Chloro-benzyl)-3-imidazol-1-ylmethyl-1H-indol...)
Affinity DataIC50:  54nMAssay Description:In vitro inhibition of human Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50127282(7-[(4-Chloro-phenyl)-imidazol-1-yl-methyl]-1-ethyl...)
Affinity DataIC50:  55nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50075004(1-Ethyl-3-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50:  57nMAssay Description:In vitro inhibition of human Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50127279(1-Ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50:  62nMAssay Description:In vitro inhibitiion of cytochrome P450 19A1 from human placental microsomes with 2.5 uM [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50127286(1-Ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50:  62nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50127285(5-Chloro-1-ethyl-7-[(4-fluoro-phenyl)-imidazol-1-y...)
Affinity DataIC50:  63nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50127281(7-[(4-Bromo-phenyl)-imidazol-1-yl-methyl]-1-ethyl-...)
Affinity DataIC50:  70nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50075002(5-Bromo-3-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50:  79nMAssay Description:In vitro inhibition of human Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50127280(5-Bromo-1-ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl...)
Affinity DataIC50:  90nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50127283(7-[(3-Chloro-phenyl)-imidazol-1-yl-methyl]-1-ethyl...)
Affinity DataIC50:  110nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50127284(7-[(3-Chloro-phenyl)-imidazol-1-yl-methyl]-1-ethyl...)
Affinity DataIC50:  170nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50127287(5-Bromo-1-ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl...)
Affinity DataIC50:  200nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50075005(1-Ethyl-5-(imidazol-1-yl-phenyl-methyl)-1H-indole ...)
Affinity DataIC50:  205nMAssay Description:In vitro inhibition of human Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50075007(5-Bromo-1-ethyl-2-[(4-fluoro-phenyl)-imidazol-1-yl...)
Affinity DataIC50:  238nMAssay Description:In vitro inhibition of human Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50127278(1-Ethyl-7-[(4-fluoro-phenyl)-[1,2,4]triazol-1-yl-m...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM50075006(3-(Imidazol-1-yl-phenyl-methyl)-1-(toluene-4-sulfo...)
Affinity DataIC50:  5.40E+3nMAssay Description:In vitro inhibition of human Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Nantes University

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)
Affinity DataIC50:  2.98E+4nMAssay Description:Inhibition of CYP19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank