Affinity DataIC50: 6nMAssay Description:Inhibition of GST-fused CDK5/p25 expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of GST-fused CDK5/p25 expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of GST-fused CDK5/p25 expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using myelin protein and [33P-gamma]-ATP after 30 mins by scintillation ...More data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of GST-fused CDK5/p25 expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 119nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of GST-fused CDK5/p25 expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 137nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 147nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 149nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of GST-fused CDK5/p25 expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of GST-fused CDK5/p25 expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 and [33P-gamma]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of GST-fused CDK5/p25 expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using myelin protein and [33P-gamma]-ATP after 30 mins by scintillation ...More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using myelin protein and [33P-gamma]-ATP after 30 mins by scintillation ...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of GST-fused CDK5/p25 expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using myelin protein and [33P-gamma]-ATP after 30 mins by scintillation ...More data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using myelin protein and [33P-gamma]-ATP after 30 mins by scintillation ...More data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 and [33P-gamma]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 and [33P-gamma]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate and [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using myelin protein and [33P-gamma]-ATP after 30 mins by scintillation ...More data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibition of GST-fused CDK5/p25 expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 576nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair