Affinity DataKi: 0.339nM ΔG°: -54.1kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.407nM ΔG°: -53.6kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 1nM ΔG°: -51.4kJ/mole EC50: 2nMpH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 2nM ΔG°: -49.7kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.6kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nM ΔG°: -47.9kJ/mole EC50: 16nMpH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 4nM ΔG°: -47.9kJ/mole EC50: 8nMpH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 6nM ΔG°: -46.9kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH4R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 6nM ΔG°: -46.9kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH4R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nM ΔG°: -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH4R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 32nM ΔG°: -42.8kJ/mole EC50: 79nMpH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 33nM ΔG°: -42.7kJ/mole EC50: 200nMpH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 40nM ΔG°: -42.2kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 41nM ΔG°: -42.2kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 56nM ΔG°: -41.4kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 89nM ΔG°: -40.2kJ/mole EC50: 79nMpH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 155nM ΔG°: -38.9kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 162nM ΔG°: -38.8kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair