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Found 115 with Last Name = 'lee' and Initial = 'ce'
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076285(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  1.30nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076294(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  1.90nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076292(1-Methyl-piperidine-4-carboxylic acid {(2S,3S)-3-[...)
Affinity DataKi:  2nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076291(1-Methyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  2nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076285(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  3nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076294(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  4nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076287(1-Methyl-piperidine-4-carboxylic acid [(2S,3S)-3-(...)
Affinity DataKi:  4.10nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076293(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  4.30nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM8019(2-(3-chlorophenoxy)-N-[(2S,3S)-3-hydroxy-4-{N-[2-(...)
Affinity DataKi:  4.30nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076293(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  4.80nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076291(1-Methyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  5.80nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076288(CHEMBL284955 | Piperidine-4-carboxylic acid [(2S,3...)
Affinity DataKi:  9nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076292(1-Methyl-piperidine-4-carboxylic acid {(2S,3S)-3-[...)
Affinity DataKi:  9.80nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076286(CHEMBL34051 | N-(2-Benzo[1,3]dioxol-5-yl-ethyl)-N-...)
Affinity DataKi:  15nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076287(1-Methyl-piperidine-4-carboxylic acid [(2S,3S)-3-(...)
Affinity DataKi:  58nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM8019(2-(3-chlorophenoxy)-N-[(2S,3S)-3-hydroxy-4-{N-[2-(...)
Affinity DataKi:  63nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50076288(CHEMBL284955 | Piperidine-4-carboxylic acid [(2S,3...)
Affinity DataKi:  71nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076289(CHEMBL32997 | N-((1S,2S)-3-{(2-Benzo[1,3]dioxol-5-...)
Affinity DataKi:  100nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076286(CHEMBL34051 | N-(2-Benzo[1,3]dioxol-5-yl-ethyl)-N-...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of California

Curated by ChEMBL
LigandPNGBDBM50076290(CHEMBL284151 | N-(2-Benzo[1,3]dioxol-5-yl-ethyl)-N...)
Affinity DataKi:  300nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthranilate phosphoribosyltransferase(Mycobacterium tuberculosis)
University of Auckland

LigandPNGBDBM93073(ACS No 172)
Affinity DataKi:  1.50E+3nMAssay Description:The initial screen was performed in a 96-well plate using the fluoresence-based assay previously described. An enzyme-coupled absorbance-based assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthranilate phosphoribosyltransferase(Mycobacterium tuberculosis)
University of Auckland

LigandPNGBDBM93074(ACS No 142)
Affinity DataKi:  6.30E+3nMAssay Description:The initial screen was performed in a 96-well plate using the fluoresence-based assay previously described. An enzyme-coupled absorbance-based assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthranilate phosphoribosyltransferase(Mycobacterium tuberculosis)
University of Auckland

LigandPNGBDBM93075(ACS No 145)
Affinity DataKi:  1.50E+4nMAssay Description:The initial screen was performed in a 96-well plate using the fluoresence-based assay previously described. An enzyme-coupled absorbance-based assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthranilate phosphoribosyltransferase(Mycobacterium tuberculosis)
University of Auckland

LigandPNGBDBM93076(ACS No 174)
Affinity DataKi:  1.80E+4nMAssay Description:The initial screen was performed in a 96-well plate using the fluoresence-based assay previously described. An enzyme-coupled absorbance-based assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthranilate phosphoribosyltransferase(Mycobacterium tuberculosis)
University of Auckland

LigandPNGBDBM93077(ACS No 179)
Affinity DataKi:  1.90E+4nMAssay Description:The initial screen was performed in a 96-well plate using the fluoresence-based assay previously described. An enzyme-coupled absorbance-based assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthranilate phosphoribosyltransferase(Mycobacterium tuberculosis)
University of Auckland

LigandPNGBDBM93078(ACS No 126)
Affinity DataKi:  6.00E+4nMAssay Description:The initial screen was performed in a 96-well plate using the fluoresence-based assay previously described. An enzyme-coupled absorbance-based assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthranilate phosphoribosyltransferase(Mycobacterium tuberculosis)
University of Auckland

LigandPNGBDBM93079(ACS No 165)
Affinity DataKi:  7.90E+4nMAssay Description:The initial screen was performed in a 96-well plate using the fluoresence-based assay previously described. An enzyme-coupled absorbance-based assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthranilate phosphoribosyltransferase(Mycobacterium tuberculosis)
University of Auckland

LigandPNGBDBM85513(ACS No 10 | CAS_54-21-7 | NSC_5900 | Sodium salicy...)
Affinity DataKi:  1.19E+5nMAssay Description:The initial screen was performed in a 96-well plate using the fluoresence-based assay previously described. An enzyme-coupled absorbance-based assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105306(CHEMBL3597782)
Affinity DataIC50:  32nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105310(CHEMBL3597786)
Affinity DataIC50:  43nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105280(CHEMBL3597780)
Affinity DataIC50:  87nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105308(CHEMBL3597784)
Affinity DataIC50:  97nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105278(CHEMBL3597778)
Affinity DataIC50:  108nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105276(CHEMBL3597698)
Affinity DataIC50:  112nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105274(CHEMBL3597696)
Affinity DataIC50:  195nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105268(CHEMBL3597690)
Affinity DataIC50:  248nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105272(CHEMBL3597694)
Affinity DataIC50:  314nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105310(CHEMBL3597786)
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of HIF-2alpha in human Hep3B cells assessed as downregulation of EPO mRNA expression by RT-PCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105270(CHEMBL3597692)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105308(CHEMBL3597784)
Affinity DataIC50:  1.01E+4nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B S304M mutant (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105274(CHEMBL3597696)
Affinity DataIC50:  1.59E+4nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B S304M mutant (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105307(CHEMBL3597783)
Affinity DataIC50:  2.23E+4nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105280(CHEMBL3597780)
Affinity DataIC50:  2.39E+4nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B S304M mutant (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105273(CHEMBL3597695)
Affinity DataIC50:  2.83E+4nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibition of inter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105279(CHEMBL3597779)
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B S304M mutant (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105304(CHEMBL3597781)
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B S304M mutant (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105278(CHEMBL3597778)
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B S304M mutant (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105277(CHEMBL3597699)
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B S304M mutant (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105276(CHEMBL3597698)
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B S304M mutant (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibi...More data for this Ligand-Target Pair
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50105275(CHEMBL3597697)
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity to wild type GST-tagged HIF-2alpha PAS-B S304M mutant (240 to 350) (unknown origin) expressed in Escherichia coli assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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