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Found 119 with Last Name = 'lee' and Initial = 'mk'
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090474(CHEMBL3581710)
Affinity DataIC50:  270nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090474(CHEMBL3581710)
Affinity DataIC50:  270nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM24567((2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenylbutyrate as substrate assessed as formation of p-nitrophenol preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM24567((2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenylbutyrate as substrate preincubated for 15 mins prior substrate addition measured after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM24567((2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-...)
Affinity DataIC50:  320nMAssay Description:Inhibition of porcine pancreatic lipase pre-incubated for 15 mins before p-nitrophenylbutyrate substrate addition by microplate reader based methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090504(CHEMBL3581714)
Affinity DataIC50:  500nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090504(CHEMBL3581714)
Affinity DataIC50:  500nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090483(CHEMBL3581712)
Affinity DataIC50:  590nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090483(CHEMBL3581712)
Affinity DataIC50:  590nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090486(CHEMBL3581713)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090486(CHEMBL3581713)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50251013(2,4,2',4'-tetrahydroxy-3'-prenylchalcone | CHEMBL4...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenylbutyrate as substrate assessed as formation of p-nitrophenol preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50193719((S)-5,7,7'-trihydroxy-2',2'-dimethyl-6-(3-methylbu...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of porcine pancreatic lipase pre-incubated for 15 mins before p-nitrophenylbutyrate substrate addition by microplate reader based methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50193723((S)-2-(2,4-dihydroxy-5-(3-methylbut-2-enyl)phenyl)...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of porcine pancreatic lipase pre-incubated for 15 mins before p-nitrophenylbutyrate substrate addition by microplate reader based methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of human recombinant FIH1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090480(CHEMBL3581705)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090480(CHEMBL3581705)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090481(CHEMBL3581711)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090481(CHEMBL3581711)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50242015(CHEMBL518543 | Kuwanon C, 4 | kuwanon C)
Affinity DataIC50:  1.86E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenylbutyrate as substrate assessed as formation of p-nitrophenol preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090475(CHEMBL3581709)
Affinity DataIC50:  1.92E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090475(CHEMBL3581709)
Affinity DataIC50:  1.92E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A [1-973](Homo sapiens (Human))
University of Oxford

LigandPNGBDBM50193145(2-(1-chloro-4-hydroxyisoquinoline-3-carboxamido)ac...)
Affinity DataIC50: >2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4C [1-973](Homo sapiens (Human))
University of Oxford

LigandPNGBDBM50193145(2-(1-chloro-4-hydroxyisoquinoline-3-carboxamido)ac...)
Affinity DataIC50: >2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Oxford

LigandPNGBDBM50193145(2-(1-chloro-4-hydroxyisoquinoline-3-carboxamido)ac...)
Affinity DataIC50: >2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Oxford

LigandPNGBDBM50193145(2-(1-chloro-4-hydroxyisoquinoline-3-carboxamido)ac...)
Affinity DataIC50: >2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

LigandPNGBDBM50193145(2-(1-chloro-4-hydroxyisoquinoline-3-carboxamido)ac...)
Affinity DataIC50: >2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 3A(Homo sapiens (Human))
University of Oxford

LigandPNGBDBM50193145(2-(1-chloro-4-hydroxyisoquinoline-3-carboxamido)ac...)
Affinity DataIC50: >2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50381001(CHEMBL2017114)
Affinity DataIC50:  2.84E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenylbutyrate as substrate preincubated for 15 mins prior substrate addition measured after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50083074(CHEMBL3422851)
Affinity DataIC50:  2.92E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenylbutyrate as substrate assessed as formation of p-nitrophenol preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50251014(CHEMBL465881 | moracin N)
Affinity DataIC50:  2.97E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenylbutyrate as substrate assessed as formation of p-nitrophenol preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090476(CHEMBL3581708)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090476(CHEMBL3581708)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090477(CHEMBL3581707)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090477(CHEMBL3581707)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090478(CHEMBL3581706)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090478(CHEMBL3581706)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090479(CHEMBL3581704)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50090479(CHEMBL3581704)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IL6-induced STAT3 activation in human Hep3B cells after 12 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50381284(CHEMBL2018876)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenylbutyrate as substrate assessed as formation of p-nitrophenol preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50304610(3-(5-(2-methoxybenzylidene)-4-oxo-2-thioxothiazoli...)
Affinity DataIC50:  3.21E+4nMAssay Description:Inhibition of human recombinant FIH1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50304612(2-(5-((3-(4-(ethylthio)phenyl)-1-phenyl-1H-pyrazol...)
Affinity DataIC50:  3.62E+4nMAssay Description:Inhibition of human recombinant FIH1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50304617(6-((2-methoxyphenoxy)methyl)-3-(quinolin-2-yl)thia...)
Affinity DataIC50:  4.14E+4nMAssay Description:Inhibition of human recombinant FIH1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A [1-973](Homo sapiens (Human))
University of Oxford

LigandPNGBDBM103845(4HQ derivative 8)
Affinity DataIC50:  4.30E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50304614(CHEMBL594893 | N-(benzo[c][1,2,5]oxadiazol-4-yl)-2...)
Affinity DataIC50:  4.53E+4nMAssay Description:Inhibition of human recombinant FIH1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50304616(6-(2-methoxystyryl)-3-(quinolin-2-yl)thiazolo[2,3-...)
Affinity DataIC50:  4.75E+4nMAssay Description:Inhibition of human recombinant FIH1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50304613(CHEMBL593127 | N-(benzo[c][1,2,5]oxadiazol-4-yl)-3...)
Affinity DataIC50:  4.86E+4nMAssay Description:Inhibition of human recombinant FIH1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

LigandPNGBDBM103843(4HQ derivative 6)
Affinity DataIC50:  5.20E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50114928(CHEMBL3609152)
Affinity DataIC50:  5.48E+4nMAssay Description:Inhibition of porcine pancreatic lipase pre-incubated for 15 mins before p-nitrophenylbutyrate substrate addition by microplate reader based methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50083070(CHEMBL3422848)
Affinity DataIC50:  5.64E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenylbutyrate as substrate assessed as formation of p-nitrophenol preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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