TargetRhodopsin kinase GRK1(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Inhibition of rhodopsin kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 525nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
Affinity DataKi: 2.57E+3nMAssay Description:Compound was tested for serotonin receptor affinity by the displacement of [3H]- -5-HT binding to rat fundus membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.60E+3nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
Affinity DataKi: 2.69E+4nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+4nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
Affinity DataKi: 5.75E+4nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
Affinity DataKi: 5.80E+4nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 6.70E+4nMAssay Description:Inhibition of beta-adrenergic receptor kinase(unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 9.10E+3nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
Affinity DataKd: 1.40E+4nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
Affinity DataKd: 2.50E+4nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+4nMAssay Description:In vitro inhibition of Angiotensin I converting enzymeMore data for this Ligand-Target Pair
Affinity DataKd: 7.00E+4nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair