Compile Data Set for Download or QSAR
maximum 50k data
Found 663 with Last Name = 'lee' and Initial = 'yj'
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314290(3-benzyl-1-(4-bromophenyl)-1-(1-(pyridin-4-ylmethy...)
Affinity DataKi:  2nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314288(1-(1-((2-aminopyridin-4-yl)methyl)piperidin-4-yl)-...)
Affinity DataKi:  3nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230294(CHEMBL4071740)
Affinity DataKi:  4nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230211(CHEMBL4063126)
Affinity DataKi:  4.30nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKi:  6.70nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230212(CHEMBL4084776)
Affinity DataKi:  7nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314294(1-(4-bromophenyl)-1-(1-cyclopentylpiperidin-4-yl)-...)
Affinity DataKi:  7nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314296(1-(4-chlorophenyl)-1-(1-ethylpiperidin-4-yl)-3-(4-...)
Affinity DataKi:  7nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314291(3-benzyl-1-(4-bromophenyl)-1-(1-(pyridazin-4-ylmet...)
Affinity DataKi:  10nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314292(3-benzyl-1-(4-bromophenyl)-1-(1-cyclopentylpiperid...)
Affinity DataKi:  10nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230213(CHEMBL4092526)
Affinity DataKi:  14nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314293(1-(4-bromophenyl)-1-(1-cyclopentylpiperidin-4-yl)-...)
Affinity DataKi:  14nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230210(CHEMBL4090107)
Affinity DataKi:  16nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314311(1-(4-chlorophenyl)-3-(4-fluorobenzyl)-1-(1-(pyridi...)
Affinity DataKi:  16nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314295(1-(4-bromophenyl)-3-(3,4-dichlorobenzyl)-1-(1-ethy...)
Affinity DataKi:  23nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314313(1-(4-bromophenyl)-1-(1-cyclopentylpiperidin-4-yl)-...)
Affinity DataKi:  36nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314297(1-(5-chloropyridin-2-yl)-1-(1-ethylpiperidin-4-yl)...)
Affinity DataKi:  41nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314315(1-(4-bromophenyl)-1-(1-cyclopentylpiperidin-4-yl)-...)
Affinity DataKi:  47nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314289(1-(4-chlorophenyl)-3-(4-fluorobenzyl)-1-(1-(pyrida...)
Affinity DataKi:  49nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230209(CHEMBL4100272)
Affinity DataKi:  65nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314307(1-(4-bromophenyl)-3-(4-fluorobenzyl)-1-(1-(2-hydro...)
Affinity DataKi:  67nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314306(1-(4-chlorophenyl)-3-(4-fluorobenzyl)-1-(1-(2-hydr...)
Affinity DataKi:  86nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314314(1-(4-bromophenyl)-1-(1-cyclopentylpiperidin-4-yl)-...)
Affinity DataKi:  191nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314298(1-(1-ethylpiperidin-4-yl)-3-(4-fluorobenzyl)-1-(4-...)
Affinity DataKi:  447nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314300(1-(1-ethylpiperidin-4-yl)-3-(4-fluorobenzyl)-1-(4-...)
Affinity DataKi:  560nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314312(1-(4-chlorophenyl)-3-(4-fluorobenzyl)-1-(1-((2-hyd...)
Affinity DataKi:  624nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230293(CHEMBL4082253)
Affinity DataKi:  795nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314305(1-(4-chlorophenyl)-3-(4-fluorobenzyl)-1-(1-(methyl...)
Affinity DataKi:  858nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314308(1-(4-chlorophenyl)-1-(1-(2,3-dihydroxypropyl)piper...)
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314304(1-(4-chlorophenyl)-3-(4-fluorobenzyl)-1-(piperidin...)
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314310(1-(4-chlorophenyl)-3-(4-fluorobenzyl)-1-(1-(pyridi...)
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314302(1-(1-ethylpiperidin-4-yl)-3-(4-fluorobenzyl)-1-(pi...)
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314301(1-(4-bromobenzyl)-1-(1-ethylpiperidin-4-yl)-3-(4-f...)
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314299(1-(1-cyclopentylpiperidin-4-yl)-3-(4-fluorobenzyl)...)
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314309(4-(1-(4-chlorophenyl)-3-(4-fluorobenzyl)ureido)-N-...)
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314303(1-(1-ethylpiperidin-4-yl)-3-(4-fluorobenzyl)-1-(1-...)
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381743(CHEMBL2023619)
Affinity DataIC50:  0.320nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-induced IL8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381724(CHEMBL2022858)
Affinity DataIC50:  0.400nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-induced IL8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381737(CHEMBL2021945)
Affinity DataIC50:  0.5nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-induced IL8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381744(CHEMBL2023620)
Affinity DataIC50:  0.600nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-induced IL8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381733(CHEMBL2022651)
Affinity DataIC50:  0.630nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-induced IL8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381729(CHEMBL2023243)
Affinity DataIC50:  0.720nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-induced IL8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381748(CHEMBL2022656)
Affinity DataIC50:  0.890nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-induced IL8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of A disintegrin and metalloproteinase domain 9 (ADAM9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381730(CHEMBL2023244)
Affinity DataIC50:  1.06nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-induced IL8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381728(CHEMBL2023241)
Affinity DataIC50:  1.10nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-induced IL8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381749(CHEMBL2022657)
Affinity DataIC50:  1.5nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-induced IL8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362450(CHEMBL1940557)
Affinity DataIC50:  1.60nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-stimulated IL-8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381742(CHEMBL2023618)
Affinity DataIC50:  1.60nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-induced IL8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362458(CHEMBL1940694)
Affinity DataIC50:  1.69nMAssay Description:Transrepression activity at glucocorticoid receptor in human H292 cells assessed as inhibition of TNF-stimulated IL-8 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 663 total ) | Next | Last >>
Jump to: