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Found 293 with Last Name = 'levacher' and Initial = 'v'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  21.6nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  52.4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392711(CHEMBL2151380)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392710(CHEMBL2151379)
Affinity DataKi:  385nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392701(CHEMBL2151370)
Affinity DataKi:  504nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392708(CHEMBL2151377)
Affinity DataKi:  689nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392708(CHEMBL2151377)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392709(CHEMBL2151378)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392707(CHEMBL2151376)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392711(CHEMBL2151380)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392699(CHEMBL2151368)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392700(CHEMBL2151369)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392702(CHEMBL2151371)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392703(CHEMBL2151372)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392704(CHEMBL2151373)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392705(CHEMBL2151374)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392712(CHEMBL2151381)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392710(CHEMBL2151379)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392709(CHEMBL2151378)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392707(CHEMBL2151376)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392706(CHEMBL2151375)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392705(CHEMBL2151374)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392704(CHEMBL2151373)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392703(CHEMBL2151372)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392702(CHEMBL2151371)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392701(CHEMBL2151370)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392699(CHEMBL2151368)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392700(CHEMBL2151369)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392706(CHEMBL2151375)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392712(CHEMBL2151381)
Affinity DataKi:  3.64E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50291665(CHEMBL4165327)
Affinity DataIC50:  0.360nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ever...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50291432(CHEMBL4159705)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ever...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50238227(CHEMBL4071377)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of AChE in human erythrocytes using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured every mi...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured every mi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50238223(CHEMBL4102333)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of AChE in human erythrocytes using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50238216(CHEMBL4095535)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of AChE in human erythrocytes using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50449479(CHEMBL4168520)
Affinity DataIC50:  6nMAssay Description:Inhibition of human erythrocytes AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured eve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50449479(CHEMBL4168520)
Affinity DataIC50:  6nMAssay Description:Inhibition of bovine erythrocytes AChE using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50238235(CHEMBL4081915)
Affinity DataIC50:  8.80nMAssay Description:Inhibition of AChE in human erythrocytes using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50291438(CHEMBL4161065)
Affinity DataIC50:  10nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ever...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50291612(CHEMBL4163678)
Affinity DataIC50:  11nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50238224(CHEMBL4094081)
Affinity DataIC50:  14nMAssay Description:Inhibition of AChE in human erythrocytes using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50291664(CHEMBL4173239)
Affinity DataIC50:  17nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ever...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50238213(CHEMBL4066548)
Affinity DataIC50:  18nMAssay Description:Inhibition of AChE in human erythrocytes using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50291633(CHEMBL4165973)
Affinity DataIC50:  18nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ever...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50238225(CHEMBL4060011)
Affinity DataIC50:  18nMAssay Description:Inhibition of AChE in human erythrocytes using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50238212(CHEMBL4077952)
Affinity DataIC50:  20nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Vfp Therapies

Curated by ChEMBL
LigandPNGBDBM50238212(CHEMBL4077952)
Affinity DataIC50:  20nMAssay Description:Inhibition of human erythrocytes AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured eve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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