Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to human 5HT3More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Binding affinity to human 5HT3More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of Human immunodeficiency virus 1 3B proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of Human immunodeficiency virus 1 3B proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of Human immunodeficiency virus 1 3B proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of Human immunodeficiency virus 1 3B proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of Human immunodeficiency virus 1 3B proteaseMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair