TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.0350nMAssay Description:Displacement of [3H]nicotine from alpha4beta2 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]nicotine from alpha4beta2 nAChR in rat brain membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Binding affinity to alpha4beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]nicotine from alpha4beta2 nAChR in rat cerebral membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 1.33nMAssay Description:Displacement of [3H]cystisine from alpha4beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 7.60nMAssay Description:Binding affinity to alpha4beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 394nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 440nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 469nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 514nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 520nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 2.79E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nAChR in rat brain membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 2.79E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nAChR in Wistar rat hindlimb muscleMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 3.80E+3nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 5.10E+3nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 1.03E+4nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 1.13E+4nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 1.80E+4nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 2.80E+4nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 3.50E+4nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 4.00E+4nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 4.30E+4nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 4.90E+4nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 5.00E+4nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 1.84E+5nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cortical membranes by beta countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 2.77E+5nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 3.25E+5nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: >5.00E+5nMAssay Description:Displacement of [125I]-alpha-Bungarotoxin from alpha7 nAChR rat cortical membranes by gamma countingMore data for this Ligand-Target Pair