Affinity DataKi: 30nMAssay Description:Binding affinity for cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity for cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataKi: 7.50E+3nMAssay Description:Binding affinity for cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+4nMAssay Description:Binding affinity for cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 1.81E+4nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
Affinity DataIC50: 3.96E+4nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
Affinity DataIC50: 6.51E+4nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
Affinity DataIC50: 7.63E+4nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 8.10E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
Affinity DataIC50: 9.43E+4nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 9.50E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 1.03E+5nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 1.09E+5nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 1.13E+5nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
Affinity DataIC50: 1.96E+5nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: 2.34E+5nMAssay Description:Inhibitory concentration against cytochrome P450 2D6More data for this Ligand-Target Pair