Affinity DataKi: 0.150nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 147nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 579nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 635nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.52E+3nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.76E+3nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.99E+3nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 2.11E+3nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 4.40E+3nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 9.50E+3nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 2.26E+4nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:In vitro opioid receptor delta mediated mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:In vitro inhibitory activity against opioid activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 0.590nMAssay Description:In vitro inhibitory activity against opioid activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:In vitro opioid receptor delta mediated mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro opioid receptor delta mediated mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Displacement of [3H]- DPDPE from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:In vitro opioid receptor delta mediated mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:In vitro opioid receptor delta mediated mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of opioid receptor mu in guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:In vitro opioid inhibitory activity against in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Compound is tested in vitro in mouse vas deferens (MVD) assay mediated by Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Displacement of [3H]- DPDPE from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro opioid receptor delta mediated mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:In vitro opioid receptor delta mediated mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Compound is tested in vitro in mouse vas deferens (MVD) assay mediated by Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:In vitro inhibitory activity against opioid activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Displacement of [3H]- DPDPE from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:In vitro opioid inhibitory activity against in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Compound is tested in vitro in mouse vas deferens (MVD) assay mediated by Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:In vitro opioid inhibitory activity against in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Displacement of [3H]- DAGO from opioid receptor mu in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Displacement of [3H]- DPDPE from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Opioid receptor binding affinity in rat brain membrane preparations by the displacement of [3H]DSLET (Opioid receptor delta 1-selective radioligand)More data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Displacement of [3H]- DAGO from opioid receptor mu in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Evaluated for the inhibition of [3H]DAGO binding to mu-receptor of guinea pig brainMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Displacement of [3H]- DPDPE from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Evaluated for the inhibition of [3H]DAGO binding to mu-receptor of guinea pig brainMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Evaluated for the inhibition of [3H]DAGO binding to mu-receptor of guinea pig brainMore data for this Ligand-Target Pair