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Found 19 with Last Name = 'marhefka' and Initial = 'ca'
TargetAndrogen receptor(Homo sapiens (Human))
The University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM18699((2R)-3-bromo-2-hydroxy-2-methyl-N-[4-nitro-3-(trif...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against human androgen receptor (hAR) in competitive binding assayMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18665((2S)-3-(4-acetamidophenoxy)-2-hydroxy-2-methyl-N-[...)
Affinity DataKi:  3.98nM ΔG°:  -44.6kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18675((2S)-2-hydroxy-3-(4-isothiocyanatophenoxy)-2-methy...)
Affinity DataKi:  4.62nM ΔG°:  -44.2kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18661((2R)-3-[(4-acetamidophenyl)sulfanyl]-2-hydroxy-2-m...)
Affinity DataKi:  4.90nM ΔG°:  -44.1kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18667((2S)-2-hydroxy-2-methyl-N-[4-nitro-3-(trifluoromet...)
Affinity DataKi:  6.07nM ΔG°:  -43.6kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18663((2S)-3-(4-fluorophenoxy)-2-hydroxy-2-methyl-N-[4-n...)
Affinity DataKi:  6.11nM ΔG°:  -43.6kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18676((2S)-3-[(4-fluorophenyl)amino]-2-hydroxy-2-methyl-...)
Affinity DataKi:  7.96nM ΔG°:  -43.0kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18668((2S)-3-(4-chlorophenoxy)-2-hydroxy-2-methyl-N-[4-n...)
Affinity DataKi:  9.56nM ΔG°:  -42.5kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18669((2S)-3-(4-bromophenoxy)-2-hydroxy-2-methyl-N-[4-ni...)
Affinity DataKi:  11.6nM ΔG°:  -42.1kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18672((2S)-2-hydroxy-3-(4-methoxyphenoxy)-2-methyl-N-[4-...)
Affinity DataKi:  13.7nM ΔG°:  -41.7kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
The University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50099679(3-Bromo-2-hydroxy-2-methyl-N-(4-nitro-3-trifluorom...)
Affinity DataKi:  16.5nMAssay Description:Binding affinity against human androgen receptor (hAR) in competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18674((2S)-2-hydroxy-3-[4-(1H-indol-5-yl)phenoxy]-2-meth...)
Affinity DataKi:  17.0nM ΔG°:  -41.2kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18670((2S)-2-hydroxy-3-(4-iodophenoxy)-2-methyl-N-[4-nit...)
Affinity DataKi:  30.0nM ΔG°:  -39.9kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18671((2S)-2-hydroxy-2-methyl-3-(4-methylphenoxy)-N-[4-n...)
Affinity DataKi:  34.8nM ΔG°:  -39.6kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18666((2S)-3-(4-acetylphenoxy)-2-hydroxy-2-methyl-N-[4-n...)
Affinity DataKi:  36.6nM ΔG°:  -39.5kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
The University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50099680((R)-N-(4-Amino-3-trifluoromethyl-phenyl)-3-bromo-2...)
Affinity DataKi:  80.9nMAssay Description:Binding affinity against human androgen receptor (hAR) in competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18677((2S)-3-[(4-acetamidophenyl)amino]-2-hydroxy-2-meth...)
Affinity DataKi:  128nM ΔG°:  -36.6kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18664((2R)-3-(4-fluorophenoxy)-2-hydroxy-2-methyl-N-[4-n...)
Affinity DataKi:  225nM ΔG°:  -35.3kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Tennessee At Memphis

LigandPNGBDBM18673(Nonsteroidal AR Ligand, S-14 | tert-butyl N-{4-[(2...)
Affinity DataKi:  336nM ΔG°:  -34.3kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed