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Found 42 with Last Name = 'masetti' and Initial = 'm'
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114409(CHEMBL3609809)
Affinity DataKi:  3.90E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as disappearance of NADH fluorescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114409(CHEMBL3609809)
Affinity DataKi:  4.70E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using NADH as substrate assessed as disappearance of NADH fluorescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386758(CHEMBL2046893)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386758(CHEMBL2046893)
Affinity DataIC50:  2.51nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386755(CHEMBL2046889)
Affinity DataIC50:  15.8nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386755(CHEMBL2046889)
Affinity DataIC50:  17nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386757(CHEMBL2046892)
Affinity DataIC50:  39.8nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386757(CHEMBL2046892)
Affinity DataIC50:  44nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386756(CHEMBL2046890)
Affinity DataIC50:  62nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386756(CHEMBL2046890)
Affinity DataIC50:  63.1nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386760(CHEMBL2046895)
Affinity DataIC50:  192nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386760(CHEMBL2046895)
Affinity DataIC50:  200nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386753(CHEMBL2046891)
Affinity DataIC50:  580nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386753(CHEMBL2046891)
Affinity DataIC50:  631nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386754(CHEMBL2046888)
Affinity DataIC50:  2.79E+3nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386754(CHEMBL2046888)
Affinity DataIC50:  2.79E+3nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386759(CHEMBL2046894)
Affinity DataIC50:  7.86E+3nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386759(CHEMBL2046894)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114404(CHEMBL3608325)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114409(CHEMBL3609809)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114408(CHEMBL3609810)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114400(CHEMBL3608329)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114403(CHEMBL3608326)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114401(CHEMBL3608328)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114409(CHEMBL3609809)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114407(CHEMBL3197264)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114402(CHEMBL3608327)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114399(CHEMBL3608330)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114404(CHEMBL3608325)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114400(CHEMBL3608329)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114403(CHEMBL3608326)
Affinity DataIC50:  1.05E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114399(CHEMBL3608330)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114405(CHEMBL3609813)
Affinity DataIC50:  1.25E+5nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114405(CHEMBL3609813)
Affinity DataIC50:  1.34E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114412(CHEMBL3609812)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114402(CHEMBL3608327)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114401(CHEMBL3608328)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114407(CHEMBL3197264)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114408(CHEMBL3609810)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114410(CHEMBL3608332)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114411(CHEMBL3608331)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50114406(CHEMBL3609811)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed