Affinity DataIC50: 0.900nMAssay Description:Inhibition of human recombinant renin compound treated for 10 mins before substrate addition measured after 90 mins by fluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human recombinant renin compound treated for 10 mins before substrate addition measured after 90 mins by fluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human plasma renin activity after 60 mins by competitive RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human plasma renin activity after 60 mins by competitive RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Inhibition of cynomolgus monkey plasma renin activity after 60 mins by competitive RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of cynomolgus monkey plasma renin activity after 60 mins by competitive RIAMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human cathepsin EMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 54nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.40nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.80nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.5nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.5nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.40nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair